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lapatinib bevarede betydelig aktivitet over for brystcancercellelinjer selekteret for langtidsvækst i trastuzumab- holdigt medium in vitro.
lapatinib retained significant activity against breast cancer cell lines selected for long-term growth in trastuzumab-containing medium in vitro.
hiv-1-isolater med en nedsat følsomhed over for amprenavir er selekteret efter en række in vitro- passager.
hiv-1 isolates with a decreased susceptibility to amprenavir have been selected during in vitro serial passage experiments.
ritonavir-resistente isolater af hiv-1 er blevet selekteret in vitro og isoleret fra patienter i behandling med terapeutiske doser af ritonavir.
ritonavir-resistant isolates of hiv-1 have been selected in vitro and isolated from patients treated with therapeutic doses of ritonavir.
desuden er en k70e-substitution i hiv 1-reverse transkriptase blevet selekteret af tenofovir, hvilket fører til en nedsat følsomhed for tenofovir på lavt niveau.
in addition, a k70e substitution in hiv-1 reverse transcriptase has been selected by tenofovir and results in low-level reduced susceptibility to tenofovir.
disse mutationer blev selekteret hos patienter med præeksisterende raltegravir-resistens, som efterfølgende blev behandlet med dolutegravir (anført som en sekundær mutation for dolutegravir).
these mutations have been selected in patients with pre-existing raltegravir resistance and who were then treated with dolutegravir (listed as secondary mutations for dolutegravir).
bemærk: følgende varianter blev selekteret i cellekultur, men var ikke behandlingsrelaterede: ns3- varianter: a156t hos genotype 1a samt r155q og d168h hos genotype 1b.
note: the following variants were selected in cell culture but were not treatment-emergent: ns3 variants a156t in genotype 1a, and r155q and d168h in genotype 1b; ns5a variants y93c/h in genotype 1a, and l31f/v or y93h in combination with l28m, l31f/v or p58s in genotype 1b; and ns5b variants y448h in genotype 1a, and m414t and y448h in genotype 1b.
k65r-mutationen kan desuden selekteres ved hjælp af abacavir eller didanosin og forårsager nedsat følsomhed over for disse stoffer samt lamivudin, emtricitabin og tenofovir.
the k65r mutation can also be selected by abacavir or didanosine and results in reduced susceptibility to these agents plus lamivudine, emtricitabine and tenofovir.