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dasatinib hæmmer aktivitet af bcr- abl kinasen og kinaser, der tilhører src- kinasefamilien samt en række andre udvalgte onkogene kinaser, inklusive c- kit, ephrinreceptor- kinaser og pdgfβ - receptorer.
dasatinib inhibe l'activité de la kinase bcr-abl, des kinases de la famille src, d'un certain nombre d'autres kinases oncogènes sélectives dont le c-kit, des récepteurs de l'éphrine (eph), et du récepteur β du pdgf.