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bovendien wordt zaleplon gemetaboliseerd door cyp3a4 en omgezet in desethylzaleplon, dat verder wordt gemetaboliseerd door aldehyde-oxydase en dan omgezet wordt in 5-oxo-desethylzaleplon.
additionally, zaleplon is metabolised by cyp3a4 to form desethylzaleplon which is further metabolised by aldehyde oxidase to form 5-oxo-desethylzaleplon.
Last Update: 2017-04-26
Usage Frequency: 3
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zevenenvijftig procent (57%) van de dosis wordt teruggevonden in urine in de vorm van 5-oxo-zaleplon en zijn glucuronide-metaboliet, en nog eens 9% wordt teruggevonden als 5-oxo- desethylzaleplon en zijn glucuronide-metaboliet.
fifty-seven percent (57%) of the dose is recovered in urine in the form of 5-oxo-zaleplon and its glucuronide metabolite, an additional 9% is recovered as 5-oxo-desethylzaleplon and its glucuronide metabolite.
Last Update: 2017-04-26
Usage Frequency: 3
Quality: