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zowel cyp2d6 als cyp1a2 katalyseren de vorming van de twee belangrijkste metabolieten glucuronideconjugaat van 4-hydroxyduloxetine en sulfaatconjugaat van 5-hydroxy,6- methoxyduloxetine.
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Last Update: 2011-10-23
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zowel cytochroom p450-2d6 als 1a2 katalyseren de vorming van de twee belangrijkste metabolieten glucuronideconjugaat van 4-hydroxyduloxetine en sulfaatconjugaat van 5- hydroxy,6-methoxyduloxetine.
formarea celor doi metaboliţi majori, conjugatul glucuronid al 4- hidroxi- duloxetinei şi conjugatul sulfat al 5 - hidroxi, 6- metoxi- duloxetinei, este catalizată de izoenzimele citocromului p450- 2d6 şi 1a2.
Last Update: 2012-04-10
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