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norfluoxetine half-lives are increased to 7 and 12 days, respectively.
alkoholio sukelta kepen ciroze) fluoksetino ir norfluoksetino pusins eliminacijos laikas pailgja atitinkamai iki 7 ir 12 dien.
Last Update: 2008-03-04
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fluoxetine and its metabolite norfluoxetine, are known to be excreted in human breast milk.
Žindymo laikotarpis fluoksetino ir norfluoksetino prasiskverbia į motinos pieną.
Last Update: 2012-04-11
Usage Frequency: 2
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elimination the elimination half-life of fluoxetine is 4 to 6 days and for norfluoxetine 4 to16 days.
fluoksetino pusinės eliminacijos laikas yra 4- 6 dienos, norfluoksetino – 4- 16 dienų.
Last Update: 2012-04-11
Usage Frequency: 2
Quality:
fold higher than that observed in adolescents and the mean norfluoxetine concentration 1.5-fold higher.
vidutin norfluoksetino koncentracija 1, 5 karto didesn uz paaugli.
Last Update: 2008-03-04
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lactation:fluoxetine and its metabolite norfluoxetine, are known to be excreted in human breast milk.
zindymo laikotarpis fluoksetino ir norfluoksetino prasiskverbia motinos pien.
Last Update: 2008-03-04
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following the last dose administration, fluoxetine and norfluoxetine plasma levels declined steadily in a log-linear fashion.
po paskutinės dozės skyrimo fluoksetino ir norfluoksetino kiekiai kraujo plazmoje palaipsniui mažėjo ilga logaritmine tiese.
Last Update: 2012-04-11
Usage Frequency: 2
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fluoxetine is primarily metabolised by the liver to the active metabolite norfluoxetine (desmethylfluoxetine) , by desmethylation.
daugiausia fluoksetino metabolizuojama demetilinimo bdu kepenyse, susidarant aktyviam metabolitui norfluoksetinui (demetilfluoksetinui) .
Last Update: 2008-03-04
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norfluoxetine plasma levels slowly appeared in plasma and were slowly eliminated with t½ values ranging from 44.2 to 48.9 hours on day 21.
21 dieną.
Last Update: 2011-10-23
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lactation:fluoxetine and its metabolite norfluoxetine, are known to be excreted in human breast milk.adverse events have been reported in breastfeeding infants.
tokie pozymiai gali rodyti serotonino receptori suzadinim arba nutraukimo sindrom.mint simptom atsiradimo laikas ir trukm gali bti susij su ilgu fluoksetino (4-6 dienos) ir jo aktyvaus metabolito norfluoksetino (4-16 dien) pusins eliminacijos laiku.zindymo laikotarpis fluoksetino ir norfluoksetino prasiskverbia motinos pien.zindomiems kdikiams pasireisk nepageidaujam reiskini.
Last Update: 2008-03-04
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the mean fluoxetine concentration in children is approximately 2- fold higher than that observed in adolescents and the mean norfluoxetine concentration 1.5-fold higher.
vidutinė fluoksetino koncentracija vaikų organizme maždaug 2 kartus, o vidutinė norfluoksetino koncentracija – 1, 5 karto didesnė už paauglių.
Last Update: 2012-04-11
Usage Frequency: 2
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a 6-week washout interval should be observed following discontinuation of therapy with reconcile prior to the administration of any veterinary medicinal product that may adversely interact with fluoxetine or its metabolite, norfluoxetine.
prieš skiriant kitą veterinarinį vaistą po gydymo reconcile, būtina laikytis 6 sav. pasišalinimo iš organizmo laikotarpio, nes gali nepalankiai reaguoti su fluoksetinu ar jo metabolitu - norfluoksetinu.
Last Update: 2017-04-26
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as in adults, fluoxetine and norfluoxetine accumulated extensively following multiple oral dosing; steady-state concentrations were achieved within 3 to 4 weeks of daily dosing.
geriant kartotines vaistinio preparato dozes, daug fluoksetino iremea/chmp/46089/2006/lt21/63© emea 2006 norfluoksetino susikaupia kaip ir suaugusij organizme.kasdiena vartojant vaistin preparat, pusiausvyros apykaitos koncentracijos pasiekiamos per 3-4 savaites.
Last Update: 2008-03-04
Usage Frequency: 1
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the elimination half-life of fluoxetine is 4 to 6 days and for norfluoxetine 4 to16 days.these long half-lives are responsible for persistence of the drug for 5-6 weeks after discontinuation.
fluoksetino pusins eliminacijos laikas yra 4-6 dienos, norfluoksetino 4-16 dien.dl tokio ilgo pusins eliminacijos laiko vaistinis preparatas islieka organizme 5-6 savaites po to, kai baigiamas jo vartojimas.
Last Update: 2008-03-04
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at 10 mg/kg/day, plasma levels achieved in animals were approximately 0.8 to 8.8 fold (fluoxetine) and 3.6 to 23.2 fold (norfluoxetine) those usually observed in paediatric patients.
10 mg/kg kno svorio doz per par gavusi gyvn plazmoje susidar mazdaug 0, 8-8, 8 kartus (fluoksetino) ir 3, 6-23, 2 karto (norfluoksetino) didesns koncentracijos plazmoje, palyginti su prastai nustatoma vaikams ir paaugliams.
Last Update: 2008-03-04
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