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tyrimai su žmogaus kepenų mikrosomomis parodė, kad retapamulinas yra stiprus cyp3a4 inhibitorius.
in human liver microsomes, retapamulin was shown to be a strong inhibitor of cyp3a4.
Last Update: 2017-04-26
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eksperimentai in vitro su žmogaus kepenų mikrosomomis rodo, kad pirmiausiai lopinaviras metabolizuojamas oksidacijos būdu.
in vitro experiments with human hepatic microsomes indicate that lopinavir primarily undergoes oxidative metabolism.
Last Update: 2017-04-26
Usage Frequency: 1
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tyrimų su žmogaus mikrosomomis metu nustatyta, kad eltrombopago gliukuronizaciją veikia ugt1a1 ir ugt1a3 fermentai.
human liver microsome studies identified ugt1a1 and ugt1a3 as the enzymes responsible for eltrombopag glucuronidation.
Last Update: 2017-04-26
Usage Frequency: 1
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metabolizmas.eksperimentai in vitro su zmogaus kepen mikrosomomis rodo, kad pirmiausiai lopinaviras metabolizuojamas oksidacijos bdu.
metabolism: in vitro experiments with human hepatic microsomes indicate that lopinavir primarily undergoes oxidative metabolism.
Last Update: 2008-03-04
Usage Frequency: 3
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tyrimai in vitro su žmogaus kepenų mikrosomomis parodė, kad daugiausia simepreviro metabolizuojama oksidacijos būdu kepenų cyp3a4 sistemoje.
in vitro experiments with human liver microsomes indicated that simeprevir primarily undergoes oxidative metabolism by the hepatic cyp3a4 system.
Last Update: 2017-04-26
Usage Frequency: 1
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tyimai in vitro su zmogaus kepen mikrosomomis rodo, kad entakaponas slopina citochrom p450 2c9 (ic50 4 µm) .
data from in vitro studies using human liver microsomal preparations indicate that entacapone inhibits cytochrome p450 2c9 (ic50 ~ 4 µm) .
Last Update: 2008-03-04
Usage Frequency: 3
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metabolizmas in vitro eksperimentai su zmogaus kepen mikrosomomis (zkm) rodo, kad daugiausia vyksta darunaviro oksidacinis metabolizmas.
metabolism in vitro experiments with human liver microsomes (hlms) indicate that darunavir primarily undergoes oxidative metabolism.
Last Update: 2008-03-04
Usage Frequency: 1
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tyimai in vitro su žmogaus kepenų mikrosomomis rodo, kad entakaponas slopina citochromą p450 2c9 (ic50 ∼ 4 µm).
data from in vitro studies using human liver microsomal preparations indicate that entacapone inhibits cytochrome p450 2c9 (ic50 ~ 4 µm).
Last Update: 2012-04-11
Usage Frequency: 2
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tyrimai in vitro, naudojant zmogaus kepen mikrosomas, parod, kad daugiausia aprepitanto metabolizuoja cyp3a4, maziau cyp1a2 ir cyp2c19.
in vitro studies using human liver microsomes indicate that aprepitant is metabolised primarily by cyp3a4 and potentially with minor contribution by cyp1a2 and cyp2c19.
Last Update: 2008-03-04
Usage Frequency: 5
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