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dasatinibul acționează în principal prin blocarea proteinkinazei bcr-abl.
dasatinib acts mainly by blocking the bcr-abl protein kinase.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
substanţa activă din votrient, pazopanibul, este un inhibitor al proteinkinazei.
the active substance in votrient, pazopanib, is a protein kinase inhibitor.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
nilotinibul acţionează prin blocarea proteinkinazei numite kinaza „bcr-abl”.
nilotinib acts by blocking the protein kinase called bcr-abl kinase.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
dasatinib acţionează în principal prin blocarea proteinkinazei numite kinaza „ bcr - abl ”.
dasatinib acts mainly by blocking the protein kinase called ‘ bcr-abl’ kinase.
Last Update: 2012-04-11
Usage Frequency: 2
Quality:
cobimetinib este un inhibitor reversibil, selectiv, alosteric, cu administrare pe cale orală, care blochează calea proteinkinazei activate de mitogen (mapk), ţintind kinazele 1 şi 2 activate de mitogen reglate de semnale extracelulare (mek 1 şi mek 2), ceea ce determină inhibarea fosforilării kinazelor 1 şi 2 reglate de semnalul extracelular (erk 1 şi erk 2).
cobimetinib is a reversible, selective, allosteric, oral inhibitor that blocks the mitogen-activated protein kinase (mapk) pathway by targeting the mitogen-activated extracellular signal-regulated kinase (mek) 1 and mek 2 which results in inhibition of phosphorylation of the extracellular signal- regulated kinase (erk) 1 and erk 2.
Last Update: 2017-04-26
Usage Frequency: 1
Quality: