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safinamid deluje prek dopaminergičnega in nedopaminergičnega mehanizma delovanja.
safinamide acts through both dopaminergic and non-dopaminergic mechanisms of action.
Last Update: 2017-04-26
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pri nenadni prekinitvi dopaminergičnega zdravljenja so poročali o simptomih, ki kažejo na maligni nevroleptični sindrom.
symptoms suggestive of neuroleptic malignant syndrome have been reported with abrupt withdrawal of dopaminergic therapy.
Last Update: 2017-04-26
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pri raziskovanju dopaminergičnega delovanja na živalskih modelih so bili glavni presnovki 100- krat manj učinkoviti od ropinirola.
none of the many metabolites formed are involved in the resulting activity of the product and the main metabolite is 100 times less potent than ropinirole in animal models examining dopaminergic function.
Last Update: 2012-04-11
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vendar pa se opikapon uporablja kot dodatno zdravljenje k levodopi, zato je treba razmisliti o prilagajanjih odmerka na podlagi možnega povečanega dopaminergičnega odziva na levodopo in s tem povezanim prenašanjem.
however, as opicapone is to be used as adjunctive levodopa-therapy, dose adjustments may be considered based on a potentially enhanced levodopa dopaminergic response and associated tolerability.
Last Update: 2017-04-26
Usage Frequency: 1
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