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data för receptoraffinitet och mitogenicitet in vitro gav inga bevis för en ökad mitogen potential jämfört med humant insulin.
receptor affinity data and in vitro mitogenicity tests revealed no evidence of an increased mitogenic potential compared to human insulin.
Last Update: 2017-04-26
Usage Frequency: 3
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in vitro har affinitet för andra receptorer endast upptäckts i koncentrationer som minst 150-faldigt överstiger dess 5-ht4 receptoraffinitet.
in vitro, only at concentrations exceeding its 5-ht4 receptor affinity by at least 150-fold, affinity for other receptors was detected.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
i de prekliniska studierna visade olanzapin (ki <100 nm) receptoraffinitet för serotonin 5ht2a/2c, 5ht3, 5ht6; dopamin d1, d2, d3, d4, d5; kolinerga muskarinreceptorer m1-m5; α1- adrenoreceptorer och histamin-h1-receptorer.
in preclinical studies, olanzapine exhibited a range of receptor affinities (ki < 100 nm) for serotonin 5 ht2a/2c, 5 ht3, 5 ht6; dopamine d1, d2, d3, d4, d5; cholinergic muscarinic receptors m1-m5; α1 adrenergic; and histamine h1 receptors.
Last Update: 2017-04-26
Usage Frequency: 8
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