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also, less than 0.1% of the administered dose is excreted as the metabolite n-desethyloxybutynin.
inoltre, meno dello 0,1% della dose somministrata viene escreta sotto forma del metabolito n-desetil-ossibutinina.
Last Update: 2012-04-12
Usage Frequency: 3
Quality:
metabolites include phenylcyclohexylglycolic acid, which is pharmacologically inactive, and n-desethyloxybutynin, which is pharmacologically active.
i metaboliti comprendono l’acido fenilcicloesil glicolico, farmacologicamente inattivo, e la n-desetil- ossibutinina, che è farmacologicamente attiva.
Last Update: 2017-04-26
Usage Frequency: 4
Quality:
the difference in auc and cmax of oxybutynin and the active metabolite n-desethyloxybutynin following transdermal administration of kentera on either the abdomen, buttocks or hip is not clinically relevant.
la differenza dell’ auc e della cmax dell’ ossibutinina e del metabolito attivo, la n-desetil- ossibutinina, a seguito della somministrazione transdermica di kentera sull’ addome, sui glutei o sul fianco, non ha rilevanza clinica.
Last Update: 2012-04-12
Usage Frequency: 3
Quality:
the difference in auc and cmax of oxybutynin and the active metabolite n-desethyloxybutynin following transdermal administration of kentera on either the abdomen, upper arms/shoulders and thighs is not clinically relevant.
in seguito alla somministrazione transdermica di kentera sull’addome, sulla parte superiore delle braccia/spalle o sulle cosce non vi sono differenze clinicamente rilevanti nell’auc e nella cmax dell’ossibutinina e del metabolita attivo n-desetilossibutinina.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
the active metabolite, n-desethyloxybutynin, has pharmacological activity on the human detrusor muscle that is similar to that of oxybutynin in vitro studies, but has a greater binding affinity for parotid tissue than oxybutynin.
il metabolito attivo, la n-desetil- ossibutinina, ha un’ attività farmacologica sul muscolo detrusore umano simile a quella degli studi in vitro con l’ ossibutinina, ma ha un’ affinità di legame al tessuto parotideo maggiore dell’ ossibutinina.
Last Update: 2012-04-12
Usage Frequency: 3
Quality: