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Ritonavir induces CYP3A4, CYP1A2, CYP2C9 and glucuronosyl transferase.

O ritonavir induz o CYP3A4, CYP1A2, CYP2C9 e a transferase glucuronosilo.

Last Update: 2008-03-04
Subject: Medical
Usage Frequency: 2
Quality:
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Data are not available to indicate whether tipranavir inhibits or induces glucuronosyl transferases.

Não existem dados disponíveis que indiquem se o tipranavir inibe ou induz as glucoronosil tranferases.

Last Update: 2008-03-04
Subject: Medical
Usage Frequency: 2
Quality:
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Ritonavir also inhibits CYP2D6 and induces CYP3A4, CYP1A2, CYP2C9 and glucuronosyl transferase.

O ritonavir também inibe a CYP2D6 e induz a CYP3A4, CYP1A2, CYP2C9 e a transferase glucuronosilo.

Last Update: 2008-03-04
Subject: Medical
Usage Frequency: 2
Quality:
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Caution should be exercised when deferasirox is combined with strong UDP- glucuronosyl transferase (UGT) inducers, or CYP2C8 substrates (see section 4.5).
http://www.emea.europa.eu/

Deve ter- se precaução quando o deferasirox é usado em combinação com indutores potentes do UDP- glucuronosil transferase, ou substratos do CYP2C8 (ver secção 4. 5).
http://www.emea.europa.eu/

Last Update: 2012-04-12
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

Medicinal products that affect etravirine exposure Etravirine is metabolised by CYP3A4, CYP2C9 and CYP2C19 followed by glucuronidation by uridine diphosphate glucuronosyl transferase (UDPGT).
http://www.emea.europa.eu/

Medicamentos que afectam a exposição da etravirina A etravirina é metabolizada pelo CYP3A4, CYP2C9 e CYP2C19 seguida de glucoronidação efectuada pela glucoroniltransferase da uridina difosfato (UDPGT).
http://www.emea.europa.eu/

Last Update: 2012-04-12
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

Hyperbilirubinaemia Reversible elevations in indirect (unconjugated) bilirubin related to inhibition of UDP-glucuronosyl transferase (UGT) have occurred in patients receiving REYATAZ (see section 4.8).
http://www.emea.europa.eu/

Hiperbilirrubinemia Em doentes medicados com REYATAZ ocorreram elevações reversíveis da bilirrubina indirecta (não conjugada) relacionadas com a inibição da UDP- glucuronosil transferase (UGT) (ver secção 4. 8).
http://www.emea.europa.eu/

Last Update: 2012-04-12
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

Hyperbilirubinemia Reversible elevations in indirect (unconjugated) bilirubin related to inhibition of UDP-glucuronosyl transferase (UGT) have occurred in patients receiving REYATAZ (see section 4.8) .

Hiperbilirrubinemia Em doentes medicados com REYATAZ ocorreram elevações reversíveis da bilirrubina indirecta (não conjugada) relacionadas com a inibição da UDP-glucuronosil transferase (UGT) (ver secção 4. 8) .

Last Update: 2008-03-04
Subject: Medical
Usage Frequency: 5
Quality:
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