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Caution should be exercised when deferasirox is combined with strong UDP- glucuronosyl transferase (UGT) inducers, or CYP2C8 substrates (see section 4.5).
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Deve ter- se precaução quando o deferasirox é usado em combinação com indutores potentes do UDP- glucuronosil transferase, ou substratos do CYP2C8 (ver secção 4. 5).
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Last Update: 2012-04-12 |
Medicinal products that affect etravirine exposure Etravirine is metabolised by CYP3A4, CYP2C9 and CYP2C19 followed by glucuronidation by uridine diphosphate glucuronosyl transferase (UDPGT).
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Medicamentos que afectam a exposição da etravirina A etravirina é metabolizada pelo CYP3A4, CYP2C9 e CYP2C19 seguida de glucoronidação efectuada pela glucoroniltransferase da uridina difosfato (UDPGT).
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Last Update: 2012-04-12 |
Hyperbilirubinaemia Reversible elevations in indirect (unconjugated) bilirubin related to inhibition of UDP-glucuronosyl transferase (UGT) have occurred in patients receiving REYATAZ (see section 4.8).
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Hiperbilirrubinemia Em doentes medicados com REYATAZ ocorreram elevações reversíveis da bilirrubina indirecta (não conjugada) relacionadas com a inibição da UDP- glucuronosil transferase (UGT) (ver secção 4. 8).
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Last Update: 2012-04-12 |
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