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lisaks on klofarabiin vastupidavam lagundamisele rakkudes adenosiindeaminaasi toimel ja oma klassi kuuluvate teiste toimeainetega võrreldes vähem vastuvõtlik fosforolüütilisele lõhustamisele, kuid klofarabiintrifosfaadi afiinsus dna polümeraas ja ribonukleotiidreduktaasi suhtes on samasugune või suurem kui desoksüadenosiintrifosfaadil.
in addition, clofarabine possesses greater resistance to cellular degradation by adenosine deaminase and decreased susceptibility to phosphorolytic cleavage than other active substances in its class whilst the affinity of clofarabine triphosphate for dna polymerase and ribonucleotide reductase is similar to or greater than that of deoxyadenosine triphosphate.
Last Update: 2017-04-26
Usage Frequency: 1
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8 peale selle on klofarabiin vastupidavam rakkude lagundamisele adenosiindeaminaasi toimel ja oma klassi kuuluvate teiste toimeainetega võrreldes vähem vastuvõtlik fosforolüütilisele lõhustamisele, kuid klofarabiintrifosfaadi afiinsus dna polümeraas α ja ribonukleotiidreduktaasi suhtes on samasugune või suurem kui desoksüadenosiintrifosfaadil.
in addition, clofarabine possesses greater resistance to cellular degradation by adenosine deaminase and decreased susceptibility to phosphorolytic cleavage than other active substances in its class whilst the affinity of clofarabine triphosphate for dna polymerase α and ribonucleotide reductase is similar to or greater than that of deoxyadenosine triphosphate.
Last Update: 2012-04-11
Usage Frequency: 2
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