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L’ interazione potenziale tra farmaci, collegata al transporter cationico organico (OCT), tra metilnaltrexone e un OCT inibitore è stata studiata in 18 soggetti sani confrontando i profili farmacocinetici a dose singola di metilnaltrexone prima e dopo la somministrazione di dosi multiple da 400 mg di cimetidina.
http://www.emea.europa.eu/

De organische kationtransporteur(OCT) - gerelateerde geneesmiddel-geneesmiddelinteractiepotentieel tussen methylnaltrexon en een OCT remmer werd bij 18 gezonde personen onderzocht door de enkele-dosis farmacokinetische profielen van methylnaltrexon te vergelijken voor en na meervoudige doses cimetidine 400 mg.
http://www.emea.europa.eu/

Last Update: 2012-04-11
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

Negli studi clinici sitagliptin non ha alterato significativamente le farmacocinetiche di metformina, gliburide, simvastatina, rosiglitazone, warfarin, o contraccettivi orali, fornendo evidenza in vivo di una bassa propensione a causare interazioni con i substrati di CYP3A4, CYP2C8, CYP2C9, e con il trasportatore di cationi organici (OCT).
http://www.emea.europa.eu/

In klinisch onderzoek gaf sitagliptine geen wezenlijke verandering van de farmacokinetiek van metformine, glibenclamide, simvastatine, rosiglitazon, warfarine, of orale anticonceptiva, waarmee in vivo bewezen is dat sitagliptine een lage neiging heeft om interacties te veroorzaken met substraten van CYP3A4, CYP2C8, CYP2C9 en organic cationic transporter (OCT).
http://www.emea.europa.eu/

Last Update: 2012-04-11
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

Negli studi clinici sitagliptin non ha alterato significativamente la farmacocinetica di metformina, gliburide, simvastatina, rosiglitazone, warfarin, o contraccettivi orali, fornendo evidenza in vivo di una bassa propensione a causare interazioni con i substrati di CYP3A4, CYP2C8, CYP2C9, e con il trasportatore di cationi organici (OCT).
http://www.emea.europa.eu/

In klinisch onderzoek gaf sitagliptine geen wezenlijke verandering van de farmacokinetiek van metformine, glibenclamide, simvastatine, rosiglitazon, warfarine, of orale anticonceptiva, waarmee in vivo bewezen is dat sitagliptine een lage neiging heeft om interacties te veroorzaken met substraten van CYP3A4, CYP2C8, CYP2C9 en organic cationic transporter (OCT).
http://www.emea.europa.eu/

Last Update: 2012-04-11
Subject: Pharmaceuticals
Usage Frequency: 1
Quality:

-ACP/OCT product:

-ACP/OCT product:

Last Update: 2008-03-04
Subject: Legal and Notarial
Usage Frequency: 1
Quality:
Reference: Anonymous

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