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11 permezz ta ’ oat3 (ic50=160 µm) jew p- glycoprotein (sa 250 µm) f’ kon entrazzjonijiet fil- pla ma terapewtikament relevanti.
in vitro, sitagliptin did not inhibit oat3 (ic50=160 μ m) or p-glycoprotein (up to 250 μ m) mediated transport at therapeutically relevant plasma concentrations.
Last Update: 2012-04-10
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