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afoxolaner had high systemic absorption.
altækt frásog afoxolaner er mikið.
Letzte Aktualisierung: 2017-04-26
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afoxolaner / milbemycin oxime tablets
afoxolaner / milbemýsínoxím tuggutöflur
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afoxolaner is an insecticide and acaricide of the isoxazoline family.
afoxolaner er skordýraeyðandi og mítlaeyðandi efni af flokki isoxazolina.
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afoxolaner is an insecticide and acaricide belonging to the isoxazoline family.
afoxolaner er skordýraeyðandi og mítlaeyðandi efni af flokki isoxazolina.
Letzte Aktualisierung: 2017-04-26
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afoxolaner in the dog is metabolized to more hydrophilic compounds and then eliminated.
hjá hundum umbrotnar afoxolaner í vatnsæknari efni og skilst síðan út.
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afoxolaner 11.3 mg afoxolaner 28.3 mg afoxolaner 68 mg afoxolaner 136 mg
afoxolaner 11,3 mg afoxolaner 28,3 mg afoxolaner 68 mg afoxolaner 136 mg
Letzte Aktualisierung: 2017-04-26
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afoxolaner kills fleas before egg production and therefore prevents the risk of household contamination.
afoxolaner drepur flær áður en eggjaframleiðsla hefst og hindrar því hættu á mengun á heimilum.
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after oral administration in dogs, afoxolaner was shown to have high systemic absorption following administration.
eftir inntöku hjá hundum var altækt frásog afoxolaner mikið.
Letzte Aktualisierung: 2017-04-26
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in clinical studies, no serious adverse reactions were attributed to the combination of afoxolaner and milbemycin oxime.
Í klínískum rannsóknum var ekki hægt að rekja alvarlegar aukaverkanir til samsetningar afoxolaner og milbemysínoxíms.
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prolonged afoxolaner-induced hyperexcitation results in uncontrolled activity of the central nervous system and death of insects and acarines.
langvarandi yfirörvun með afoxolaner hefur í för með sér stjórnleysi á miðtaugakerfi og dauða skordýra og mítla.
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parasites need to start feeding on the host to become exposed to afoxolaner; therefore the risk of the transmission of parasite borne diseases cannot be excluded.
sníkjudýrin verða að byrja að nærast á hýslinum til þess að verða útsett fyrir afoxolaner, þar af leiðandi er ekki hægt að útiloka að sjúkdómar berist með sníkjudýrinu.
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the selective toxicity of afoxolaner between insects, acarines and mammals may be inferred by the differential sensitivity of the insects and acarines’ gaba receptors versus mammalian gaba receptors.
mismunandi eiturhrif afoxolaner hjá skordýrum, mítlum og spendýrum getur verið vegna mismunandi næmni gaba-viðtaka skordýra og mítla annars vegar og gaba-viðtaka spendýra hins vegar.
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afoxolaner is active against adult fleas as well as several tick species such as dermacentor reticulatus and d. variabilis, ixodes ricinus and i. scapularis, rhipicephalus sanguineus, amblyomma americanum and haemaphysalis longicornis.
afoxolaner er virkt gegn fullþroska flóm og nokkrum mítlategundum eins og dermacentor reticulatus og d. variabilis, ixodes ricinus og i. scapularis, rhipicephalus sanguineus, amblyomma americanum, og haemaphysalis longicornis.
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afoxolaner acts as an antagonist at ligand-gated chloride channels, in particular those gated by the neurotransmitter gamma-aminobutyric acid (gaba).
afoxolaner virkar sem loki við bindilstýrð klóríðgöng (ligand-gated chloride channels), sérstaklega þau sem stýrð eru af taugaboðefninu gammaamínósmjörsýru (gaba).
Letzte Aktualisierung: 2017-04-26
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afoxolaner acts at ligand-gated chloride channels, in particular those gated by the neurotransmitter gamma-aminobutyric acid (gaba), thereby blocking pre- and post-synaptic transfer of chloride ions across cell membranes.
afoxolaner virkar við bindilstýrð klóríðgöng (ligand-gated chloride channels), sérstaklega þau sem stýrð eru af taugaboðefninu gammaamínósmjörsýru (gaba), og hamlar þannig flutningi klóríðjóna yfir frumuhimnur framan og aftan taugamóta.
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