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som et resultat af at hæmme serotoninoptagelse forstærker fluoxetin serotonerg neurotransmission og frembringer funktionelle virkninger, der skyldes øget aktivering af serotoninreceptorer.
as a result of inhibiting serotonin uptake, fluoxetine enhances serotonergic neurotransmission and produces functional effects resulting from increased activation of serotonin receptors.
最終更新: 2017-04-26
使用頻度: 3
品質:
asenapin udviser høj affinitet for 5-ht1a-, 5-ht1b-, 5-ht2a-, 5-ht2b-, 5-ht2c-, 5-ht5-, 5-ht6- og 5-ht7-serotoninreceptorer; d2-, d3-, d4- og d1-dopaminreceptorer; α1- og α2-adrenerge receptorer samt h1-histaminreceptorer, og moderat affinitet for h2-receptorer.
asenapine exhibits high affinity for serotonin 5-ht1a, 5-ht1b, 5-ht2a, 5-ht2b, 5-ht2c, 5-ht5, 5-ht6, and 5-ht7 receptors, dopamine d2, d3, d4, and d1 receptors), α1 and α2-adrenergic receptors, and histamine h1 receptors, and moderate affinity for h2 receptors.
最終更新: 2017-04-26
使用頻度: 2
品質: