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Η λιπεγκφιλγραστίμη μεταβολίζεται μέσω ενδοκυτταρικής ή εξωκυτταρικής αποικοδόμησης από πρωτεολυτικά ένζυμα.
lipegfilgrastim is metabolised via intra- or extracellular degradation by proteolytic enzymes.
Última atualização: 2017-04-26
Frequência de uso: 1
Qualidade:
< 2,0 είναι η συγκέντρωση που πιθανόν προκαλεί σημαντική αναστολή της ενδοκυτταρικής ανάπτυξης
< 2.0 is the concentration likely to cause significant inhibition of intracellular growth
Última atualização: 2017-04-26
Frequência de uso: 1
Qualidade:
Aviso: contém formatação HTML invisível
Ο χρόνος ενδοκυτταρικής ημίσειας ζωής του τριφωσφορικού παραγώγου στα ηπατοκκύταρα είναι 17-19 ώρες in vitro.
the intracellular half life of the triphosphate in hepatocytes is 17-19 hours in vitro.
Última atualização: 2017-04-26
Frequência de uso: 5
Qualidade:
Φωσφορυλιώνεται αποτελεσματικά από κυτταρικές κινάσες στην ενεργή τριφωσφορική μορφή, η οποία έχει χρόνο ενδοκυτταρικής ημιζωής 14 ώρες.
it is efficiently phosphorylated by cellular kinases to the active triphosphate form, which has an intracellular half-life of 14 hours.
Última atualização: 2017-04-26
Frequência de uso: 4
Qualidade:
Αποδείχθηκε ότι η πιρλιµυκίνη συγκεντρώνεται στα πολυµορφοπύρηνα κύτταρα. ∆εν αποδείχθηκε όµως η δυνατότητα ενδοκυτταρικής καταστροφής του staplylococcus aureus
pirlimycin has been shown to accumulate in polymorphonuclear cells, however, intracellular killing of staphylococcus aureus was not demonstrated.
Última atualização: 2012-04-11
Frequência de uso: 2
Qualidade:
Πρώτον, µε την αναστρέψιµη και ειδική ανταγωνιστική αναστολή της αναγωγάσης hmg- coa, επιτυγχάνει µέτρια µείωση της σύνθεσης ενδοκυτταρικής χοληστερόλης.
this results in an increase in the number of ldl-receptors on cell surfaces and enhanced receptor-mediated catabolism and clearance of circulating ldl-cholesterol.
Última atualização: 2012-04-11
Frequência de uso: 2
Qualidade:
Ενδοκυτταρική φαρμακοκινητική
intracellular pharmacokinetics
Última atualização: 2017-04-26
Frequência de uso: 8
Qualidade: