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rilpivirin deluje tako, da nekompetitivno zavira reverzno transkriptazo hiv-1.
rilpivirine activity is mediated by non-competitive inhibition of hiv-1 reverse transcriptase (rt).
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 1
Kalite:
8 reverzno transkriptazo hbv, odporen hbv pa ima tudi zmanjšano sposobnost replikacije v celični kulturi.
resistance is mediated by reduced inhibitor binding to the altered hbv reverse transcriptase, and resistant hbv exhibits reduced replication capacity in cell culture.
Son Güncelleme: 2012-04-11
Kullanım Sıklığı: 4
Kalite:
emtricitabintrifosfat in tenofovirdifosfat kompetitivno zavirata reverzno transkriptazo hiv-1, kar povzroči terminacijo verige dna.
emtricitabine triphosphate and tenofovir diphosphate competitively inhibit hiv-1 reverse transcriptase, resulting in dna chain termination.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 3
Kalite:
emtricitabin trifosfat in tenofovir difosfat kompetitivno inhibirata hiv- 1 reverzno transkriptazo, kar rezultira v prekinitvi verige dna.
emtricitabine triphosphate and tenofovir diphosphate competitively inhibit hiv-1 reverse transcriptase, resulting in dna chain termination.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 4
Kalite:
odpornost se razvije zaradi zmanjšane vezave inhibitorjev na spremenjeno reverzno transkriptazo hbv, odporen hbv pa ima tudi zmanjšano sposobnost replikacije v celični kulturi.
resistance is mediated by reduced inhibitor binding to the altered hbv reverse transcriptase, and resistant hbv exhibits reduced replication capacity in cell culture.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 3
Kalite:
veže se direktno na reverzno transkriptazo in blokira od rna in dna odvisne učinke dna- polimeraze, tako da razgradi katalitičo mesto encima.
nevirapine binds directly to reverse transcriptase and blocks the rna-dependent and dna-dependent dna polymerase activities by causing a disruption of the enzyme's catalytic site.
Son Güncelleme: 2011-10-23
Kullanım Sıklığı: 1
Kalite:
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emtricitabin trifosfat zavira podvajanje hiv z vgraditvijo v virusno dna z reverzno transkriptazo (rt) hiv, kar povzroči prekinitev verige dna.
emtricitabine triphosphate inhibits hiv replication through incorporation into viral dna by the hiv reverse transcriptase (rt), which results in dna chain-termination.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 1
Kalite:
vsaka od teh zdravilnih učinkovin, znanih kot protiretrovirusna zdravila, zavira encim (reverzno transkriptazo), ki je nujen za razmnoževanje virusa.
each of these active substances, also known as antiretroviral medicines, work by interfering with an enzyme (reverse transcriptase) that is essential for the virus to multiply.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 3
Kalite:
tenofovir difosfat zavira reverzno transkriptazo virusa hiv-1 in polimerazo virusa hbv z direktno kompeticijo za vezavo z naravnim dezoksiribonukleotidnim substratom in potem, ko je vključen v dna, povzroči prekinitev njene sinteze.
tenofovir diphosphate inhibits hiv-1 reverse transcriptase and the hbv polymerase by direct binding competition with the natural deoxyribonucleotide substrate and, after incorporation into dna, by dna chain termination.
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 3
Kalite:
lamivudin-tp, karbovir-tp (aktivna trifosfatna oblika abakavirja) in zidovudin-tp so substrati za reverzno transkriptazo (rt) virusa hiv in tudi njeni kompetitivni inhibitorji.
lamivudine-tp, carbovir-tp (the active triphosphate form of abacavir) and zidovudine-tp are substrates for and competitive inhibitors of hiv reverse transcriptase (rt).
Son Güncelleme: 2017-04-26
Kullanım Sıklığı: 3
Kalite: