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o-desmethylvenlafaxine measurement
medición de o - desmetilvenlafaxina
Last Update: 2014-12-09
Usage Frequency: 1
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o-desmethylvenlafaxine measurement (procedure)
medición de o - desmetilvenlafaxina
Last Update: 2014-12-09
Usage Frequency: 1
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imipramine did not affect the pharmacokinetics of venlafaxine and o-desmethylvenlafaxine.
imipramina no alteró las farmacocinéticas de venlafaxina ni de o− desmetilvenlafaxina.
Last Update: 2012-04-10
Usage Frequency: 2
Quality:
venlafaxine and its active metabolite, o-desmethylvenlafaxine, are excreted in breast milk.
venlafaxina y su metabolito activo o-desmetilvenlafaxina se excretan en la leche materna.
Last Update: 2012-04-10
Usage Frequency: 4
Quality:
diazepam does not appear to affect the pharmacokinetics of either venlafaxine or o-desmethylvenlafaxine.
diazepam no parece afectar la farmacocinética tanto de venlafaxina como de o- desmetilvenlafaxina.
Last Update: 2012-04-10
Usage Frequency: 4
Quality:
metoprolol did not alter the pharmacokinetic profile of venlafaxine or its active metabolite, o-desmethylvenlafaxine.
el metoprolol no alteró el perfil farmacocinético de la venlafaxina o de su metabolito activo, o-desmetilvenlafaxina.
Last Update: 2012-04-10
Usage Frequency: 2
Quality:
venlafaxine is extensively metabolised, primarily to the active metabolite, o-desmethylvenlafaxine (odv).
venlafaxina se metaboliza ampliamente, principalmente al metabolito activo o-desmetilvenlafaxina (odv).
Last Update: 2012-04-10
Usage Frequency: 2
Quality:
in vitro and in vivo studies indicate that venlafaxine is metabolised to a minor, less active metabolite, n-desmethylvenlafaxine, by cyp3a4.
los estudios in vitro e in vivo indican que venlafaxina se metaboliza a un metabolito secundario, menos activo, n-desmetilvenlafaxina, mediante cyp3a4.
Last Update: 2011-10-23
Usage Frequency: 1
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preclinical studies have shown that venlafaxine and its major metabolite, o-desmethylvenlafaxine (odv), are inhibitors of serotonin and noradrenaline reuptake.
estudios preclínicos han mostrado que venlafaxina y su metabolito principal, o-desmetilvenlafaxina (odv), son inhibidores de la recaptación de serotonina y noradrenalina.
Last Update: 2012-04-10
Usage Frequency: 2
Quality:
ketoconazole (cyp3a4 inhibitor) a pharmacokinetic study with ketoconazole in cyp2d6 extensive (em) and poor metabolisers (pm) resulted in higher auc of venlafaxine (70% and 21% in cyp2d6 pm and em subjects, respectively) and o-desmethylvenlafaxine (33% and 23% in cyp2d6 pm and em subjects, respectively) following administration of ketoconazole.
un estudio farmacocinético con ketoconazol en metabolizadores lentos (ml) y rápidos (mr) de cyp2d6 dio como resultado un auc superior de venlafaxina (del 70% y del 21% en pacientes ml y mr de cyp2d6, respectivamente) y o-desmetilvenlafaxina (del 33% y del 23% en pacientes ml y mr de cyp2d6, respectivamente) tras la administración de ketoconazol.
Last Update: 2012-04-10
Usage Frequency: 2
Quality: