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perindoprilat
perindoprilato
Last Update: 2018-03-04
Usage Frequency: 10
Quality:
perindopril acts through its active metabolite, perindoprilat.
el perindopril actúa a través de su metabolito activo, el perindoprilato.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
* dialysis clearance of perindoprilat is 70 ml/ min.
* la depuración del perindoprilato durante la diálisis es de 70 ml/ min.
Last Update: 2012-04-10
Usage Frequency: 2
Quality:
dialysis clearance of perindoprilat is equal to 70 ml/ min.
la depuración del perindoprilato durante la diálisis corresponde a 70 ml/ min.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
the peak plasma concentration of perindoprilat is achieved within 3 to 4 hours.
la concentración plasmática máxima del perindoprilato se alcanza en 3 a 4 horas.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
in addition to active perindoprilat, perindopril yields five metabolites, all inactive.
además del perindoprilato activo, el perindopril da cinco metabolitos, todos ellos inactivos.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
2 mg on the day of dialysis * dialysis clearance of perindoprilat is 70 ml/min.
2 mg en el día de la diálisis * la depuración del perindoprilato durante la diálisis es de 70 ml/min.
Last Update: 2008-03-04
Usage Frequency: 3
Quality:
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elimination of perindoprilat is decreased in the elderly, and also in patients with heart or renal failure.
la eliminación del perindoprilato disminuye entre los ancianos y entre los pacientes con insuficiencia cardíaca o renal.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
about 20% of the total quantity of perindopril absorbed is converted into perindoprilat, the active metabolite.
aproximadamente el 20% de todo el perindopril absorbido se transforma en perindoprilato, el metabolito activo.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
as ingestion of food decreases conversion to perindoprilat, hence bioavailability , should be administered orally in a single daily dose in the morning before a meal.
como la ingesta reduce la conversión hacia el perindoprilato y, por ende, la biodisponibilidad, deben administrarse por vía oral en una sola toma matutina diaria, antes del desayuno.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
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protein binding is slight (binding of perindoprilat to angiotensin converting enzyme is less than 30%), but is concentration-dependent.
la unión a las proteínas es discreta (el perindoprilato se une en menos del 30% a la enzima conversora de la angiotensina), pero depende de la concentración.
Last Update: 2012-04-10
Usage Frequency: 5
Quality:
however, the quantity of perindoprilat formed is not reduced and therefore no dosage adjustment is required (see also sections 4.2 “ posology and method of administration” and 4.4 “ special warnings and special precautions for use”).
no obstante, la cantidad generada de perindoprilato no disminuye; por eso, no se precisa ningún ajuste posológico (véanse las secciones 4.2 “ posología y forma de administración” y 4.4 “ advertencias y precauciones especiales de empleo”).
Last Update: 2012-04-10
Usage Frequency: 5
Quality: