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Bulgarian

Основните пътища на биотрансформация са оксидативно n-деалкилиране, хидроксилиране на норборнен пръстен и s-окисление.

English

the major biotransformation pathways are oxidative n-dealkylation, hydroxylation of norbornane ring, and s-oxidation.

Last Update: 2017-04-26
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Bulgarian

Проучвания in vitro с човешки чернодробни микрозоми и човешки сДНК-експресирани цитохром p450 изоензими показват, че бортезомиб се метаболизира главно оксидативно чрез цитохром p450 ензими, 3А4, 2С19 и 1А2.

English

in vitro studies with human liver microsomes and human cdna-expressed cytochrome p450 isozymes indicate that bortezomib is primarily oxidatively metabolised via cytochrome p450 enzymes, 3a4, 2c19, and 1a2.

Last Update: 2017-04-26
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Bulgarian

Метаболизъм Проучвания in vitro с човешки чернодробни микрозоми и човешки сДНК- експресирани цитохром p450 изоензими показват, че бортезомиб се метаболизира главно оксидативно чрез цитохром p450 ензими, 3А4, 2С19 и 1А2.

English

the major metabolic pathway is deboronation to form two deboronated metabolites that subsequently undergo hydroxylation to several metabolites.

Last Update: 2011-10-23
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Bulgarian

16 Метаболизъм Глимепирид се метаболизира изцяло чрез оксидативна биотрансформация както след интравенозно, така и след перорално приложение.

English

metabolism glimepiride is completely metabolised by oxidative biotransformation after either an intravenous or oral dose.

Last Update: 2012-04-10
Usage Frequency: 4
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