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dinotefuran har en lav affinitet for pattedyrs acetylkolinreceptor-bindingssteder.
dinotefuran has a low affinity for mammalian acetylcholine receptor sites.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
der er ingen mætning af bindingssteder i koncentrationsområdet opnået ved terapeutiske doser.
there is no saturation of binding sites in the concentration range reached with therapeutic doses.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
risikoen for krydsresistens mellem efavirenz og nrtier er lille på grund af de forskellige bindingssteder og virkningsmekanisme.
the potential for cross-resistance between efavirenz and nrtis is low because of the different binding sites on the target and mechanism of action.
Last Update: 2017-04-26
Usage Frequency: 4
Quality:
data fra dyreforsøg tyder på, at amlodipin binder til både dihydropyridin og ikke - dihydropyridin- bindingssteder.
experimental data suggest that amlodipine binds to both dihydropyridine and non-dihydropyridine binding sites.
Last Update: 2012-04-11
Usage Frequency: 11
Quality:
det virker på octopamin-receptor-bindingssteder hos ektoparasitter og medfører øget nerveaktivitet og død hos insekterne.
it acts at octopamine receptor sites in ectoparasites giving rise to increased nervous activity and death of insects.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
15- 30% af udgangsværdien før første dosis og mættede cd11a til < 5% af udgangsværdien af tilgængelige cd11a- bindingssteder.
pharmacodynamic effects in studies using an initial dose of 0.7 mg/ kg followed by 11 weekly doses of 1.0 mg/ kg, efalizumab maximally reduced expression of cd11a on circulating t lymphocytes to approximately 15-30% of pre-dose baseline values and saturated cd11a to < 5% of baseline available cd11a binding sites.
Last Update: 2011-10-23
Usage Frequency: 1
Quality:
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Please delete it you feel so.
dette tyder på en minimal risiko for lægemiddel- lægemiddel interaktioner gennem fortrængning fra bindingsstederne ved samtidig indgift af andre lægemidler.
this indicates minimal risk of drug-drug interactions by displacement from binding sites during concomitant administration of other drugs.
Last Update: 2012-04-11
Usage Frequency: 7
Quality: