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risperidone has no affinity for cholinergic receptors.
risperidoonil puudub afiinsus koliinergilistesse retseptoritesse.
Last Update: 2012-04-11
Usage Frequency: 2
Quality:
quadramet has a high affinity for skeletal tissue.
quadramet on luukoe suhtes suure afiinsusega.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
asenapine has no appreciable affinity for muscarinic cholinergic receptors.
asenapiin ei seondu märkimisväärselt muskariini koliinergiliste retseptoritega.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
the peptide itself has a lower affinity for these receptors.
peptiidi enda afiinsus retseptorite suhtes on madalam.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
it has a high affinity for serotoninergic 5-ht2 and dopaminergic d2 receptors.
sellel on suur afiinsus serotoniinergilistesse 5- ht2 ja dopamiinergilistesse d2 retseptoritesse.
Last Update: 2012-04-11
Usage Frequency: 2
Quality:
abacavir and lamivudine triphosphates show significantly less affinity for host cell dna polymerases.
abakaviir- ja lamivudiintrifosfaadi afiinsus peremeesorganismi dna-polümeraasi suhtes on oluliselt väiksem.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
tasimelteon exhibits a greater affinity for the mt2 as compared to the mt1 receptor.
tasimelteoonil on suurem afiinsus mt2-retseptori kui mt1-retseptori suhtes.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
ritonavir also has a high affinity for p-glycoprotein and may inhibit this transporter.
ritonaviiril on tugev afiinsus ka p-glükoproteiini suhtes ja ta võib selle transporteri aktiivsust inhibeerida.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
abacavir, lamivudine and zidovudine triphosphates show significantly less affinity for host cell dna polymerases.
lamivudiin-, abakaviir- ja zidovudiintrifosfaadi afiinsus peremeesorganismi dna-polümeraasi suhtes on oluliselt väiksem.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
the selective action of bisphosphonates on bone is based on their high affinity for mineralised bone.
bisfosfonaatide selektiivne toime luudele põhineb nende suurel afiinsusel mineraliseerunud luu suhtes.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
olanzapine demonstrated a greater in vitro affinity for serotonin 5ht2 than dopamine d2 receptors and greater
olansapiini korral esines suurem in vitro afiinsus serotoniini 5ht2 kui dopamiini d2- retseptorite suhtes ja suurem 5ht2 - kui d2- aktiivsus in vivo.
Last Update: 2011-10-23
Usage Frequency: 1
Quality:
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telmisartan does not show affinity for other receptors, including at2 and other less characterised at receptors.
telmisartaan ei ole afiinne teiste retseptorite suhtes, kaasaarvatud at2 ja teised vähemtuntud at-retseptorid.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
ethanol's affinity for water can lead to problems with the product's final quality.
etanooli afiinsuse tõttu vee suhtes võib langeda lõpptoote kvaliteet.
Last Update: 2017-04-06
Usage Frequency: 1
Quality:
both losartan and its principal active metabolite have a far greater affinity for the at1 receptor than for the at2 receptor.
nii losartaanil kui aktiivsel põhimetaboliidil on palju suurem afiinsus at1 - kui at2- retseptorite suhtes.
Last Update: 2012-04-11
Usage Frequency: 4
Quality:
it weakly inhibits dopamine reuptake with no significant affinity for histaminergic, dopaminergic, cholinergic and adrenergic receptors.
ta inhibeerib vähesel määral dopamiini tagasihaaret ning omab mitteolulist afiinsust histamiinergiliste, dopamiinergiliste, kolinergiliste ja adrenergiliste retseptorite suhtes.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
ulipristal acetate also has high affinity for the glucocorticoid receptor and in vivo, in animals, antiglucocorticoid effects have been observed.
ulipristaalatsetaadil on suur afiinsus ka glükokortikoidretseptori suhtes ja in vivo on loomadel täheldatud glükokortikoidide vastast toimet.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
olanzapine demonstrated a greater in vitro affinity for serotonin 5ht2 than dopamine d2 receptors and greater 5ht2 than d2 activity in vivo models.
olansapiini korral esines suurem in vitro afiinsus serotoniini 5ht2 kui dopamiini d2-retseptorite suhtes ja suurem 5ht2- kui d2-aktiivsus in vivo.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
the binding of strontium to human plasma proteins is low (25%) and strontium has a high affinity for bone tissue.
strontsium seondub inimeste plasmavalkudega vähesel määral (25%) ja strontsiumil on luukoe suhtes suur afiinsus.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
clofarabine has high affinity for one of the activating phosphorylating enzymes, deoxycytidine kinase, which exceeds that of the natural substrate, deoxycytidine.
klofarabiinil on kõrge afiinsus ühe fosforüleerimist aktiveeriva ensüümi desoksütsütidiinkinaasi suhtes, mis ületab loodusliku substraadi desoksütsütidiini oma.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
venlafaxine has virtually no affinity for rat brain muscarinic, cholinergic, h1-histaminergic or α 1-adrenergic receptors in vitro.
venlafaksiinil ei ole in vitro olulist afiinsust roti aju muskariini -, h1- histaminergiliste ega α1 - adrenergiliste retseptorite suhtes.
Last Update: 2012-04-11
Usage Frequency: 2
Quality: