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pharmacotherapeutic group: macrolides, lincosamides and streptogramins, atc code:
atc kood:
Last Update: 2011-10-23
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this is often referred to as mlsb resistance as it affects macrolides, lincosamides and streptogramins.
sellele viidatakse sageli kui mls resistentsusele ning see hõlmab makroliide, linkosamiide ja streptogrammiine.
Last Update: 2017-04-26
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5.1 pharmacodynamic properties lon pharmacotherapeutic group: macrolides, lincosamides and streptogramins, atc code:
atc kood:
Last Update: 2011-10-23
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generally, cross-resistance between tildipirosin and other macrolides, lincosamides or streptogramins is to be expected.
Üldiselt on ootuspärane, et tildipirosiini ja teiste makroliidide, linkosamiinide või streptogramiinide vahel tekib ristresistentsus.
Last Update: 2017-04-26
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whereas that could make it necessary to use streptogramins as therapeutic agents of last resort to treat germs which have developed resistance to other antibiotics;
seetõttu võib tekkida vajadus kasutada raviainena streptogramiini kui viimast abinõu nende haigusetekitajate vastu, mis on omandanud resistentsuse muude antibiootikumide suhtes;
Last Update: 2014-11-21
Usage Frequency: 2
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whereas two streptogramins are clinically important in human medicine in the treatment of last resort of vancomycin resistant enterococci, namely pristinamycin and the combination dalfopristin/quinupristin;
vankomütsiiniresistentsete enterokokkide vastase viimase abinõuna on inimmeditsiinis kliiniliselt olulised kaks streptogramiini, nimelt pristinamütsiin ja kombineeritud ravim dalfopristiin/kinupristiin;
Last Update: 2014-11-21
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resistance to macrolides can develop by mutations in genes encoding ribosomal rna (rrna) or some ribosomal proteins; by enzymatic modification (methylation) of the 23s rrna target site, generally giving rise to cross-resistance with lincosamides and group b streptogramins (mlsb resistance); by enzymatic inactivation; or by macrolide efflux.
4 resistentsus makroliidide suhtes võib areneda ribosoomi rnad kodeerivate geenide või mõnede ribosoomivalkude mutatsiooniga; ribosoomi rna 23s sihtkoha ensümaatilise modifikatsiooniga (metülatsiooniga), mis annab tavaliselt ristresistentsuse linkoosamiidide ja b grupi streptogramiinidega (mlsb resistentsus); ensümaatilise inaktiveerimisega või makroliidi väljavoolu tõttu.
Last Update: 2012-04-11
Usage Frequency: 4
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