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inhibition of cyp isoforms
inhibícia cyp izoforiem
Last Update: 2017-04-26
Usage Frequency: 1
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cyp isoforms selective substrates:
4 selektívne substráty izoforiem cyp:
Last Update: 2012-04-12
Usage Frequency: 2
Quality:
two isoforms, cox-1 and cox-2 have been identified.
identifikovali sa dve izoformy, cox- 1 a cox- 2.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
two isoforms, cox-1 and cox-2, have been identified.
boli identifikované dve izoformy, cox- 1 a cox- 2.
Last Update: 2012-04-12
Usage Frequency: 2
Quality:
there are two isoforms of cox, cox-1, and cox-2.
cox má dve izoformy, cox-1 a cox-2.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
rivaroxaban neither inhibits nor induces any major cyp isoforms like cyp3a4.
rivaroxaban neinhibuje ani neindukuje žiadne významné izoformy cyp ako cyp3a4.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
it binds with high affinity to the vegf-a isoforms (e.g.
viaže sa s vysokou afinitou na izoformy vegf-a (napr.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
the cyclo-oxygenase enzyme (cox) is present in two isoforms.
enzým cyklo-oxygenáza (cox) existuje v dvoch formách.
Last Update: 2017-04-26
Usage Frequency: 1
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this is predominantly via cytochrome p450 2c8 although other isoforms may be involved to a lesser
metabolizmus pioglitazón sa rozsiahle metabolizuje v pečeni hydroxyláciou alifatických metylénových skupín, k čomu dochádza prevažne prostredníctvom cytochrómov p450 2c8, hoci v malom rozsahu sa týchto procesov môžu zúčastniť aj iné izoformy.
Last Update: 2011-10-23
Usage Frequency: 1
Quality:
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this is predominantly via cytochrome p450 2c8 although other isoforms may be involved to a lesser degree.
k tomu dochádza prevažne prostredníctvom cytochrómu p450 2c8, hoci v malom rozsahu sa týchto procesov môžu zúčastniť aj iné izoformy.
Last Update: 2017-04-26
Usage Frequency: 3
Quality:
based on in vitro studies, empagliflozin does not inhibit, inactivate, or induce cyp450 isoforms.
na základe štúdií in vitro empagliflozín neinhibuje, neinaktivuje ani neindukuje izoformy cyp450.
Last Update: 2017-04-26
Usage Frequency: 1
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cyp1a and cyp3a-related enzymes were identified as the feline isoforms involved in the hepatic biotransformation of maropitant.
v rámci biotransformácie maropitantu v pečeni boli u mačiek identifikované dve izoformy: cyp1a a cyp3a.
Last Update: 2017-04-26
Usage Frequency: 1
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it is unlikely that atosiban inhibits hepatic cytochrome p450 isoforms in humans (see section 4.5).
je nepravdepodobné, že atosiban inhibuje izoformy cytochrómu p450 v pečeni u ľudí (pozri časť 4.5).
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
in vitro evaluation indicated that trifluridine and fty had no inductive effect on human cyp isoforms (see section 5.2).
hodnotenie in vitro preukázalo, že trifluridín a fty nemajú indukčný vplyv na ľudské izoformy cyp (pozri časť 5.2).
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
vardenafil is metabolised predominantly by hepatic enzymes via cytochrome p450 (cyp) isoform 3a4, with some contribution from cyp3a5 and cyp2c isoforms.
vardenafil je primárne metabolizovaný pečeňovými enzýmami cez izoformu 3a4 cytochrómu p450 (cyp) s čiastočným prispením izoforiem cyp3a5 a cyp2c.
Last Update: 2017-04-26
Usage Frequency: 1
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sildenafil is a weak inhibitor of the cytochrome p450 isoforms 1a2, 2c9, 2c19, 2d6, 2e1 and 3a4 (ic50 > 150 µm).
sildenafil je slabým inhibítorom (ic50 > 150 µmol/l) izoforiem 1a2, 2c9, 2c19, 2d6, 2e1 a 3a4 cytochrómu p450.
Last Update: 2017-04-26
Usage Frequency: 1
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biotransformation tadalafil is predominantly metabolised by the cytochrome p450 (cyp) 3a4 isoform.
31 biotransformácia tadalafil sa metabolizuje najmä prostredníctvom izoformy 3a4 cytochrómu p450 (cyp).
Last Update: 2012-04-12
Usage Frequency: 4
Quality: