Results for hüdroksüleeritud translation from Estonian to English

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hüdroksüleeritud

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Estonian

uriinis tuvastati ka kaks metaboliiti (dealküleeritud ja hüdroksüleeritud metaboliidid).

English

two metabolites (a dealkylated and a hydroxylated metabolite) were also identified in urine.

Last Update: 2017-04-26
Usage Frequency: 1
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Estonian

rohkem kui 80% uriini radioaktiivsusest moodustus hüdroksüleeritud metaboliitide glükuroniidsetest konjugaatidest.

English

greater than 80 % of the radioactivity in urine was made up of glucuronide conjugates of hydroxylated metabolites.

Last Update: 2017-04-26
Usage Frequency: 3
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Estonian

osateroonatsetaat lammutub oma peamiseks - 15-hüdroksüleeritud metaboliidiks, mis on farmakoloogiliselt samuti aktiivne.

English

osaterone acetate is converted to its main, 15-hydroxylated metabolite, which is also pharmacologically active.

Last Update: 2017-04-26
Usage Frequency: 1
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Estonian

peamised metabolismiteed koertel hõlmavad metüülasendajate hüdroksüleerimist ja edasist oksüdeerimist karboksüülhappeks või hüdroksüleeritud ravimi o-glükuroniseerimist.

English

the major metabolic routes in dogs are hydroxylation of a methyl substituent and further oxidation to a carboxylic acid or o-glucuronidation of the hydroxylated product.

Last Update: 2017-04-26
Usage Frequency: 1
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Estonian

muutumatul kujul mitotaani ei ole leitud ei sapist ega uriinist, kus valdavaks on o,p’-dda koos mitmete selle hüdroksüleeritud metaboliitidega.

English

no unchanged mitotane has been found in bile or in urine, where o,p’-dda predominates, together with several of its hydroxylated metabolites.

Last Update: 2017-04-26
Usage Frequency: 3
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Estonian

inimese plasmas on kindlaks tehtud valdekoksiibi hüdroksüleeritud metaboliit (cyp tee kaudu), mis toimib cox-2 inhibiitorina.

English

a hydroxylated metabolite of valdecoxib (via the cyp pathway) has been identified in human plasma that is active as a cox-2 inhibitor.

Last Update: 2017-04-26
Usage Frequency: 3
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Estonian

biotransformatsioon: uuringud inimestel ja in vitro uuringud inimese maksa mikrosoomidega on näidanud, et efavirens metaboliseerub peamiselt tsütokroom p450 süsteemis hüdroksüleeritud metaboliitideks, millele järgneb nende metaboliitide glükuroniseerimine.

English

biotransformation: studies in humans and in vitro studies using human liver microsomes have demonstrated that efavirenz is principally metabolised by the cytochrome p450 system to hydroxylated metabolites with subsequent glucuronidation of these hydroxylated metabolites.

Last Update: 2012-04-11
Usage Frequency: 2
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Estonian

nevirapiini metaboliidid: inimese maksa mikrosoomide uuringud näitasid, et nevirapiini hüdroksüleeritud metaboliitide tekkimist ei mõjutanud dapsooni, rifabutiini, rifampitsiini ja trimetoprim/sulfametoksasooli juuresolek.

English

nevirapine metabolites: studies using human liver microsomes indicated that the formation of nevirapine hydroxylated metabolites was not affected by the presence of dapsone, rifabutin, rifampicin, and trimethoprim/sulfamethoxazole.

Last Update: 2017-04-26
Usage Frequency: 1
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Estonian

biotransformatsioon ja eliminatsioon: inimese in vivo ja inimese maksa mikrosoomide in vitro uuringud on näidanud, et nevirapiini biotransformeeritaks ulatuslikult tsütokroom p450 (oksüdatiivse) metabolismi kaudu mitmeteks hüdroksüleeritud metaboliitideks.

English

biotransformation and elimination: in vivo studies in humans and in vitro studies with human liver microsomes have shown that nevirapine is extensively biotransformed via cytochrome p450 (oxidative) metabolism to several hydroxylated metabolites.

Last Update: 2017-04-26
Usage Frequency: 1
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