Results for mikrosoomidega translation from Estonian to English

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Estonian

in vitro uuringutes inimese maksa mikrosoomidega täheldati ensüümide cyp1a2 ja cyp2b6 kerget inhibitsiooni.

English

in in vitro studies in human hepatic microsomes, minor inhibition of cyp1a2 and cyp2b6 was observed.

Last Update: 2017-04-26
Usage Frequency: 1
Quality:

Estonian

in vitro katsed inimese maksa mikrosoomidega näitavad, et darunaviir läbib põhiliselt oksüdatiivse metabolismi.

English

in vitro experiments with human liver microsomes (hlms) indicate that darunavir primarily undergoes oxidative metabolism.

Last Update: 2017-04-26
Usage Frequency: 1
Quality:

Estonian

metabolism in vitro katsed inimese maksa mikrosoomidega näitavad, et darunaviir läbib põhiliselt oksüdatiivse metabolismi.

English

metabolism in vitro experiments with human liver microsomes (hlms) indicate that darunavir primarily undergoes oxidative metabolism.

Last Update: 2012-04-11
Usage Frequency: 2
Quality:

Estonian

loomkatsed ja samuti in vitro eksperimendid inimese maksa mikrosoomidega näitasid, et ritonaviir läbis peamiselt oksüdatiivse metabolismi.

English

animal studies as well as in vitro experiments with human hepatic microsomes indicated that ritonavir primarily underwent oxidative metabolism.

Last Update: 2017-04-26
Usage Frequency: 3
Quality:

Estonian

inimese maksa mikrosoomidega teostatud in vitro uuringutes leiti, et montelukasti metabolismis osalevad tsütokroom p450 3a4, 2a6 ja 2c9.

English

in vitro studies using human liver microsomes indicate that cytochrome p450 3a4, 2a6 and 2c9 are involved in the metabolism of montelukast.

Last Update: 2012-04-11
Usage Frequency: 2
Quality:

Estonian

in vitro metabolismi uuringud inimese maksa mikrosoomidega näitasid, et cyp3a4 on peamine cyp isovorm, mis osaleb tipranaviiri metabolismis.

English

in vitro metabolism studies with human liver microsomes indicated that cyp3a4 is the predominant cyp isoform involved in tipranavir metabolism.

Last Update: 2017-04-26
Usage Frequency: 3
Quality:

Estonian

deksrasoksaani in vitro uuringutes inimese mikrosoomidega on ilmnenud deksrasoksaani suur stabiilsus, mis näitab, et põhimetabolism tsütokroom p450 kaudu on ebatõenäoline.

English

in-vitro studies on dexrazoxane in human microsomes have shown high stability of dexrazoxane indicating that major metabolism via cytochrome p450 is unlikely.

Last Update: 2017-04-26
Usage Frequency: 1
Quality:

Estonian

biotransformatsioon: inimesel ja in vitro uuringutes inimese maksa mikrosoomidega on näidatud, et atasanaviir metaboliseerub peamiselt cyp3a4 isosüümi vahendusel oksügeniseeritud metaboliitideks.

English

metabolism: studies in humans and in vitro studies using human liver microsomes have demonstrated that atazanavir is principally metabolised by cyp3a4 isozyme to oxygenated metabolites.

Last Update: 2017-04-26
Usage Frequency: 1
Quality:

Estonian

in vitro inhibeerimisuuringud inimese maksa mikrosoomidega näitavad, et tsüt okroom p450 (cyp) 1a2, 2c19 ja 3a4 osalevad leflunomiidi biotransformatsioonis.

English

in vitro inhibit ion studies in human liver microsomes suggest that cytochrome p450 (cyp) 1a2, 2c19 and 3a4 are involved in leflunomide metabolism.

Last Update: 2017-04-26
Usage Frequency: 1
Quality:

Estonian

in vitro testid inimese mikrosoomidega näitavad, et samaaegne ravi koos ainetega, mida metaboliseerivad cyp450 isovormid, võib põhjustada kas masitiniibi või nende ainete suuremaid või väiksemaid sisaldusi plasmas.

English

in vitro tests with human microsomes demonstrate that concomitant treatment with substances which are metabolised by cyp450 isoforms may result in higher or lower plasma levels of either masitinib or those substances.

Last Update: 2017-04-26
Usage Frequency: 2
Quality:

Estonian

in vitro uuringud inimese maksa mikrosoomidega on näidanud, et pemetrekseed ei põhjusta oletatavasti cyp3a, cyp2d6, cyp2c9 ja cyp1a2 poolt metaboliseeritavate ravimite metaboolse kliirensi kliiniliselt olulist vähenemist.

English

results from in vitro studies with human liver microsomes indicated that pemetrexed would not be predicted to cause clinically significant inhibition of the metabolic clearance of drugs metabolised by cyp3a, cyp2d6, cyp2c9, and cyp1a2.

Last Update: 2017-04-26
Usage Frequency: 3
Quality:

Estonian

in vitro uuringud maksa segatud mikrosoomidega, viitavad sellele, et naatriumoksübaat ei inhibeeri märkimisväärselt inimese isoensüümide aktiivsust (vt lõik 5.2).

English

studies in vitro with pooled human liver microsomes indicate that sodium oxybate does not significantly inhibit the activities of the human isoenzymes (see section 5.2).

Last Update: 2017-04-26
Usage Frequency: 3
Quality:

Estonian

in vitro uuringud inimese maksa mikrosoomidega näitavad, et tigetsükliin ei pärsi metabolismi, mis toimub konkureeriva inhibeerimise teel ühe järgmise tsütokroom p450 (cyp) isovormi vahendusel kuuest:

English

in vitro studies in human liver microsomes indicate that tigecycline does not inhibit metabolism mediated by any of the following 6 cytochrome p450 (cyp) isoforms:

Last Update: 2012-04-11
Usage Frequency: 2
Quality:

Estonian

in vitro uuringutest inimese maksa mikrosoomidega on ilmnenud, et ertapeneem ei inhibeeri kuue põhilise cyp isovormi (1a2, 2c9, 2c19, 2d6, 2e1 ja 3a4) poolt vahendatud metabolismi.

English

1a2, 2c9, 2c19, 2d6, 2e1 and 3a4.

Last Update: 2011-10-23
Usage Frequency: 1
Quality:

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