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mapk
proteínas quinasas activadas por mitógeno
Last Update: 2014-12-09
Usage Frequency: 1
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mapk p38
proteina quinasa activada por mitógeno p38
Last Update: 2014-12-09
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mapk-p44
quinasa 1 regulada por señal extracelular
Last Update: 2014-12-09
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phosphatase mapk
fosfatasa 1 de especificidad dual
Last Update: 2014-12-09
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mapk-kinases
pamqqs
Last Update: 2014-12-09
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cascade des mapk
cascada de quinasas pam
Last Update: 2014-12-09
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mapk-erk kinases
meqs
Last Update: 2014-12-09
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protéine p97(mapk)
proteína quinasa activada por mitógeno 6
Last Update: 2014-12-09
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phosphatase-1 des mapk
fosfatasa 1 de especificidad dual
Last Update: 2014-12-09
Usage Frequency: 2
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kinase-5 mapk-erk
map quinasa quinasa 5
Last Update: 2014-12-09
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mapk-erk kinase kinases
qqems
Last Update: 2014-12-09
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système de signalisation des mapk
sistema de señalización de quinasas pam
Last Update: 2014-12-09
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mapk-erk-kinase-kinase-3
map quinasa quinasa quinasa 3
Last Update: 2014-12-09
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mapk-kinase-2 régulée par des signaux extracellulaires
map quinasa quinasa 2
Last Update: 2014-12-09
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en conséquence, le cobimetinib bloque la prolifération cellulaire induite par la voie mapk en inhibant le noeud de signalisation mek1/2.
por lo tanto, cobimetinib bloquea la proliferación de células inducida por la ruta de la mapk mediante la inhibición de la señalización a nivel de mek1/2.
Last Update: 2017-04-26
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dans les modèles précliniques, l’association de cobimetinib au vemurafenib a montré que cibler simultanément les protéines braf v600 mutées et mek des cellules du mélanome inhibait la réactivation de la voie mapk par l’intermédiaire de mek1/2, conduisant au renforcement de l’inhibition du signal intracellulaire et à la diminution de la prolifération des cellules tumorales.
en los modelos preclínicos, la combinación de cobimetinib y vemurafenib mostró que la acción simúltanea sobre las proteínas brafv600 mutadas y las proteínas mek en las células del melanoma, la combinación de los dos productos que inhiben la reactivación de la ruta mapk a través de mek1/2, provoca una mayor inhibición de la señalización intracelular y una disminución de la proliferación de las células tumorales.
Last Update: 2017-04-26
Usage Frequency: 1
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