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cor pulmonale, defekt i tricuspidalklaff, hjertesvikt, kardiomegali, sinus-arrest, supraventrikulære ekstrasystoler
cardiac failure, cardiomegaly, cor pulmonale, sinus arrest, supraventricular extrasystoles, tricuspid valve incompetence
vinflunin bindes til tubulin ved eller i nærheten av vinkabindesetene og hemmer polymerisering til mikrotubuli, som resulterer i hemming av tråddannelse, forstyrrelse av mikrotubulidynamikk, mitotisk arrest og apoptose.
vinflunine binds to tubulin at or near to the vinca binding sites inhibiting its polymerisation into microtubules, which results in treadmilling suppression, disruption of microtubule dynamic, mitotic arrest and apoptosis.
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date of incorporation
Last Update: 2021-05-19
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