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metabolizare febuxostatul este metabolizat în proporţie mare prin conjugare prin sistemul enzimatic uridină difosfat glucuronoziltransferază (udpgt) şi prin oxidare prin sistemul citocromului p450
11 metabolism febuxostat is extensively metabolized by conjugation via uridine diphosphate glucuronosyltransferase (udpgt) enzyme system and oxidation via the cytochrome p450 (cyp) system.
Last Update: 2011-10-23
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febuxostatul este metabolizat în proporţie mare prin conjugare prin sistemul enzimatic uridină difosfat glucuronoziltransferază (udpgt) şi prin oxidare prin sistemul citocromului p450 (cyp).
febuxostat is extensively metabolized by conjugation via uridine diphosphate glucuronosyltransferase (udpgt) enzyme system and oxidation via the cytochrome p450 (cyp) system.
Last Update: 2017-04-26
Usage Frequency: 1
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administrarea isentress concomitent cu inductori puternici ai uridin difosfat glucuronoziltransferazelor (ugt) 1a1 (de exemplu rifampicină) trebuie făcută cu precauţie.
caution should be used when co-administering isentress with strong inducers of uridine diphosphate glucuronosyltransferase (ugt) 1a1 (e.g., rifampicin).
Last Update: 2017-04-26
Usage Frequency: 3
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