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În studiile preclinice enzalutamida nu a prezentat activitate agonistă pe receptorii androgenici.
in preclinical studies enzalutamide lacks androgen receptor agonist activity.
Last Update: 2017-04-26
Usage Frequency: 1
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are afinitate minimă pentru receptorii androgenici şi nu are afinitate pentru receptorii estrogenici sau mineralocorticoizi umani.
it has minimal affinity to the androgen receptor and no affinity for the human estrogen or mineralocorticoid receptors.
Last Update: 2017-04-26
Usage Frequency: 1
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se leagă de receptorii androgenici fără activarea exprimării genice şi, astfel, inhibă stimularea androgenică.
it binds to androgen receptors without activating gene expression and thus inhibits androgen stimulation.
Last Update: 2012-04-11
Usage Frequency: 2
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enzalutamida este un inhibitor potent al semnalizării la nivelul receptorilor androgenici care blochează câteva etape din calea de semnalizare la nivelul receptorului androgenic.
enzalutamide is a potent androgen receptor signalling inhibitor that blocks several steps in the androgen receptor signalling pathway.
Last Update: 2017-04-26
Usage Frequency: 1
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