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toceranib hämmar selektivt tyrosinkinasaktiviteten hos flera olika tyrosinkinasreceptorer, där vissa är delaktiga i tumörtillväxten, den patologiska angiogenesen och metastasprogressionen vid cancer.
toceranib selectively inhibits the tyrosine kinase activity of several members of the split kinase receptor tyrosine kinase (rtk) family some of which are implicated in tumour growth, pathologic angiogenesis, and metastatic progression of cancer.
Last Update: 2017-04-26
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tasigna är en potent hämmare av abl- tyrosinkinasaktiviteten hos bcr- abl- onkoprotein, både i cellinjer och i primära philadelphiakromosompositiva leukemiceller.
tasigna is a potent inhibitor of the abl tyrosine kinase activity of the bcr-abl oncoprotein both in cell lines and in primary philadelphia-chromosome positive leukaemia cells.
Last Update: 2012-04-11
Usage Frequency: 2
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