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kopolymer polyethylentereftalátu, hydroxylovaného polybutadienu, anhydridu pyromelové kyseliny
(polyethylene terephthalate, hydroxylated polybutadiene, pyromellitic anhydride) copolymer
Ultimo aggiornamento 2014-11-21
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v plazmě byly detekovány tři metabolity lasofoxifenu: přímý konjugát glukuronidu, glukuronid hydroxylovaného metabolitu a metylovaný katechol.
three metabolites of lasofoxifene were detected in plasma: the direct glucuronide conjugate, the glucuronide of a hydroxylated metabolite, and the methylated catechol.
Ultimo aggiornamento 2017-04-26
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diastereomer hydroxylovaného derivátu, n-glukuronidu indakaterolu, a c- a n-dealkylované produkty byly dalšími nalezenými metabolity.
a diastereomer of the hydroxylated derivative, a n-glucuronide of indacaterol, and c- and n-dealkylated products were further metabolites identified.
Ultimo aggiornamento 2017-04-26
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současné podávání duloxetinu (40 mg dvakrát denně) zvyšuje hodnotu rovnovážné (steady- state) auc tolterodinu (2 mg dvakrát denně) o 71 %, ale neovlivňuje farmakokinetiku jeho aktivního 5- hydroxylovaného metabolitu; úprava dávky není nutná.
the co-administration of duloxetine (40 mg twice daily) increases steady state auc of tolterodine (2 mg twice daily) by 71 %, but does not affect the pharmacokinetics of its active 5- hydroxyl metabolite and no dosage adjustment is recommended.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 5
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