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additionally, in various organs pharmacodynamically mediated atrophy of epithelia was observed in both species.
lisaks täheldati mõlema liigi korral eri elundites farmakodünaamiliselt vahendatud epiteeli atroofiat.
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roflumilast is extensively metabolised in humans, with the formation of a major pharmacodynamically active metabolite, roflumilast n-oxide.
roflumilast metaboliseerub inimestel olulisel määral farmakodünaamiliselt aktiivseks põhimetaboliidiks roflumilast n-oksiidiks.
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however, the predicted amount of metabolite accumulation at steady state is not pharmacodynamically important because the terminal elimination half-life is only 1–2 hours in these subjects.
metaboliit siiski ei kogune püsikontsentratsiooni juures farmakodünaamiliselt olulises koguses, sest terminaalse eliminatsiooni poolväärtusaeg on neil uuringualustel üksnes 1…2 tundi.
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the pharmacodynamically predictable and most commonly reported adverse reactions are thirst, dry mouth and pollakiuria occurring in approximately 18%, 9% and 6% of patients.
farmakodünaamiliselt ennustatavateks ja kõige sagedasemateks kõrvaltoimeteks olid janu, suukuivus ja pollakisuuria, mis esinesid ligikaudu 18%-l, 9%-l ja 6%-l patsientidest.
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the pharmacodynamically predictable and most commonly reported adverse reactions are thirst, polyuria, nocturia, and pollakiuria occurring in approximately 55%, 38%, 29% and 23% of patients, respectively.
farmakodünaamiliselt prognoositavad ja kõige sagedamini esinevad kõrvaltoimed on janu, polüuuria, noktuuria ja pollakisuuria, mida esineb vastavalt ligikaudu 55%, 38%, 29% ja 23% patsientidest.
Ultimo aggiornamento 2017-04-26
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