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Inglese

Francese

Informazioni

Inglese

zso lo no1 raciborz event type:

Francese

zso lo no1 raciborz type d'événement:

Ultimo aggiornamento 2015-05-14
Frequenza di utilizzo: 1
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Inglese

hello zso, how are you? tell me what is your mood today?

Francese

hello szo, comment vas-tu ? quelle est ton humeur du jour ?

Ultimo aggiornamento 2018-02-13
Frequenza di utilizzo: 1
Qualità:

Inglese

i had that fantastic opportunity talking with new-york art director and illustrator zso.

Francese

j’ai eu la super opportunité de m’entretenir avec zso, directrice artistique et illustratrice new-yorkaise.

Ultimo aggiornamento 2018-02-13
Frequenza di utilizzo: 1
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Inglese

a compound of formula (i), or a pharmaceutically acceptable salt, hydrate, complex or pro-drug thereof, wherein one of r1 and r2 is h, and the other is selected from c1-8-alkyl, c3-6-cycloalkyl and c1-8-alkyl-c5-10-aryl; r3 is selected from tert-butylmethyl, zso-propylmethyl, sec- butyl, tert-butyl, cyclopentyl, cyclohexyl and 1-methylcyclopentyl; r9 is selected from the following: wherein: r4 is selected from c1-8-alkyl and c3-8-cycloalkyl; g is selected from: ) ch, ) cme and n; e is selected from: o, s, ) so2, )nh, )nme and n-oxide ()n->o); j and r are independently selected from: )ch, n and n-oxide ()n-^o); and r41 is selected from amino, methylamino, dimethylamino, isopropylamino, isopropyl(methyl)amino, cyclopropylamino, cyclopropyl(methyl)amino, cyclopentylamino, morpholino, piperidin-1-yl, piperidin-1-ylmethyl, morpholinomethyl, 4-methylpiperazin-l-yl, 4-(2-methoxyethyl)piperazin-l-yl, 1- moφholinoethyl, l-(dimethylamino)ethyl, l-(methylamino)ethyl, 4-fluoro-l- methylpyrrolidin-2-yl, 4,4-difluoropiperidin-l-yl, piperidin-4-yl, l-methylpiperidin-4- yl, pyridin-3-ylamino, pyridin-2-ylamino, l-methylpyrrolidin-3-yl, methyl, isopropyl. the invention further relates to pharmaceutical compositions comprising compounds of formula (i), and the use of such compounds in the treatment of various diseases.

Francese

l'invention porte sur un composé de formule (i), ou sur un sel, un hydrate, un complexe ou un promédicament pharmaceutiquement acceptable de celui-ci. dans la formule, r1 ou r2 représente h et r2 ou r1 est choisi parmi alkyle en c1-8, cycloalkyle en c3-6 et alkyl en c1-8-aryle en c5-10; r est choisi parmi tert-butylméthyle, isopropylméthyle, sec- butyle, tert-butyle, cyclopentyle, cyclohexyle et 1-méthylcyclopentyle; r est choisi parmi ce qui suit : où : r4 est choisi parmi alkyle en c1-8 et cycloalkyle en c3-8; g est choisi parmi : )ch, )cme et n; e est choisit parmi o, s, ) so2, )nh, )nme et n-oxyde ()n->o); j et r sont choisis indépendamment parmi : )ch, n et n-oxyde ()n-^o); et r41 est choisi parmi amino, méthylamino, diméthylamino, isopropylamino, isopropyl(méthyl)amino, cyclopropylamino, cyclopropyl(méthyl)amino, cyclopentylamino, morpholino, pipéridin-1-yle, pipéridin-1-ylméthyle, morpholinométhyle, 4-méthylpipérazin-l-yle, 4-(2-méthoxyéthyl)pipérazin-l-yle, 1- morpholinoéthyle, l-(diméthylamino)éthyle, l-(méthylamino)éthyle, 4-fluoro-l-méthylpyrrolidin-2-yle, 4,4-difluoropipéridin-l-yle, pipéridin-4-yle, l-méthylpipéridin-4-yle, pyridin-3-ylamino, pyridin-2-ylamino, l-méthylpyrrolidin-3-yle, méthyle, isopropyle. l'invention porte également sur des compositions pharmaceutiques comprenant des composés de formule (i) et sur l'utilisation de ces composés dans le traitement de diverses maladies.

Ultimo aggiornamento 2011-07-27
Frequenza di utilizzo: 1
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