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lanolin, hydroxylated
lanolīns, hidroksilēts
Ultimo aggiornamento 2014-11-07
Frequenza di utilizzo: 1
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glycerides, milk, hydroxylated
glicerīdi, piena, hidroksilēti
Ultimo aggiornamento 2014-11-07
Frequenza di utilizzo: 1
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there are several hydroxylated metabolites of quinidine.
hinidīnam ir vairāki hidroksilēti metabolīti.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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authorising isopropyl ester of the hydroxylated analogue of methionine
ar ko atļauj metionīna hidroksilētā analoga izopropilesteri
Ultimo aggiornamento 2014-10-23
Frequenza di utilizzo: 1
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a hydroxylated derivative was the most prominent metabolite in serum.
nozīmīgākais metabolīts serumā bija hidroksilētais atvasinājums.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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unchanged emodepside and hydroxylated derivatives are the major excretion products.
neizmainīts edmodepsīds un hidroksilēti atvasinājumi ir galvenie ekskrēcijas produkti.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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(polyethylene terephthalate, hydroxylated polybutadiene, pyromellitic anhydride) copolymer
(polietilēna tereftalāta, hidroksilēta polibutadiēna, piromelītskābes anhidrīda) kopolimērs
Ultimo aggiornamento 2014-11-21
Frequenza di utilizzo: 1
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ketoconazole and erythromycin significantly inhibited the formation of nevirapine hydroxylated metabolites.
ketokonazols un eritromicīns būtiski inhibē nevirapīna hidroksilēto metabolītu veidošanos.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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phenolic o-glucuronides of indacaterol and hydroxylated indacaterol were further prominent metabolites.
nākamie pamanāmākie metabolīti bija indakaterola fenola o-glikuronīdi un hidroksilētais indakaterols.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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faecal excretion predominates with unchanged emodepside and hydroxylated derivatives as the major excretion products.
ar fekālijām edmodepsīds tiek izvadīts galvenokārt neizmainītā un hidroksilētu atvasinājumu veidā.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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oxidative metabolism catalysed by cyp3a4 and cyp2c8 leads to the formation of hydroxylated and dealkylated products.
oksidatīvā metabolisma ceļā ar katalizatoriem cyp3a4 un cyp2c8 tiek panākta hidroksilētu un dealkilētu produktu veidošanās.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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greater than 80 % of the radioactivity in urine was made up of glucuronide conjugates of hydroxylated metabolites.
vairāk nekā 80 % radioaktivitātes urīnā nodrošināja hidroksilēto metabolītu glikuronīda konjugāti.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 6
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osaterone acetate is converted to its main, 15-hydroxylated metabolite, which is also pharmacologically active.
osaterona acetāts pārveidojas galvenajā 15- hidroksilāta metabolītā, kas arī ir farmakoloģiski aktīvs.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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the major metabolites, hydroxylated and demethylated agomelatine, are not active and are rapidly conjugated and eliminated in the urine.
galvenie metabolīti, kas rodas agomelatīnam hidroksilējoties un demetilējoties, nav aktīvi un ātri konjugējas un izdalās ar urīnu.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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the formation of these hydroxylated metabolites is catalysed by cyp2c8, cyp3a4, and both cyp2c8 and cyp3a4 isoenzymes, respectively.
Šo hidroksilēto metabolītu veidošanos katalizē attiecīgi cyp2c8, cyp3a4 un gan cyp2c8, gan cyp3a4 izoenzīmi.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 1
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hepatic metabolism of norelgestromin occurs and metabolites include norgestrel, which is largely bound to shbg, and various hydroxylated and conjugated metabolites.
norelgestromīns metabolizējas aknās un tā metabolītos ietilpst norgestrels, kas plaši piesaistās shbg, un dažādi hidroksilēti un konjugēti metabolīti.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
Qualità:
based on in vitro studies, saquinavir is rapidly metabolised to a range of mono- and di-hydroxylated inactive compounds.
Ņemot vērā in vitro pētījumu rezultātus, sakvinavīrs tiek ātri metabolizēts par mono-un dihidroksilētiem neaktīviem savienojumiem.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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three metabolites of lasofoxifene were detected in plasma: the direct glucuronide conjugate, the glucuronide of a hydroxylated metabolite, and the methylated catechol.
plazmā konstatēti trīs lazofoksifēna metabolīti: tiešie glikuronīda konjugāti, hidroksilēto metabolītu glikuronīdi un metilētie kateholi.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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a hydroxylated metabolite of valdecoxib (via the cyp pathway) has been identified in human plasma that is active as a cox-2 inhibitor.
cilvēka plazmā konstatēts hidroksilēts valdekoksiba metabolīts (veidojas ar cyp saistītajā metabolisma ceļā), kurš izrādās aktīvs cox-2 inhibitors.
Ultimo aggiornamento 2017-04-26
Frequenza di utilizzo: 3
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biotransformation: studies in humans and in vitro studies using human liver microsomes have demonstrated that efavirenz is principally metabolised by the cytochrome p450 system to hydroxylated metabolites with subsequent glucuronidation of these hydroxylated metabolites.
biotransformācija: pētījumi cilvēkiem un in vitro pētījumi, izmantojot aknu mikrosomas, ir pierādījuši, ka efavirenzu galvenokārt metabolizē citohroma p450 sistēma līdz hidroksilētiem metabolītiem ar sekojošu šo metabolītu glikuronidēšanu.
Ultimo aggiornamento 2012-04-10
Frequenza di utilizzo: 2
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