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additionally, dasatinib inhibits src family kinases at subnanomolar concentrations.
barra minn hekk, dasatinib jinibixxi l- kinasi tal- familja src f' koncentrazzjoni subnanomolari.
these non-clinical studies show that dasatinib can overcome imatinib resistance resulting from bcr-abl overexpression, bcr-abl kinase domain mutations, activation of alternate signaling pathways involving the src family kinases (lyn, hck), and multidrug resistance gene overexpression.
13 imatinib li jirriżulta minn espressjoni żejda ta ’ bcr- abl, mutazzjonijiet fid- domain tal- kinase bcr - abl, attivazzjoni ta 'passaġġi tas- sinjalazzjoni alternattivi li jinvolvu l- kinasi tal- familja src (lyn, hck), u espressjoni żejda tal- ġene tar- reżistenza għal ħafna mediċini.