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tādējādi dctf intracelulārās koncentrācijas samazināšanās veicina dfdctf iekļaušanos dns.
thus, the reduced intracellular concentration of dctp potentiates the incorporation of dfdctp into dna.
Ultimo aggiornamento 2012-04-10
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otrkārt, dfdctf konkurē ar dctf par iekļaušanos dns (pašpotencēšana).
second, dfdctp competes with dctp for incorporation into dna (self-potentiation).
Ultimo aggiornamento 2012-04-10
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gemcitabīna citotoksisko darbību nosaka dfdcdf un dfdctf divu darbību izraisīta dns sintēzes kavēšana.
the cytotoxic effect of gemcitabine is due to inhibition of dna synthesis by two mechanisms of action by dfdcdp and dfdctp.
Ultimo aggiornamento 2012-04-10
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dfdctf farmakokinētika Šis metabolīts ir atrodams perifērisko asiņu mononukleārās šūnās un turpmāk norādītā informācija attiecas uz šīm šūnām.
dfdctp kinetics this metabolite can be found in peripheral blood mononuclear cells and the information below refers to these cells.
Ultimo aggiornamento 2012-04-10
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ja gemcitabīna koncentrācija plazmā pārsniedz 5 µg/ ml, dfdctf līmenis nepalielinās, kas liecina, ka tā sintēzei šajās šūnās ir piesātinošs raksturs.
at gemcitabine plasma concentrations above 5 µg/ml, dfdctp levels do not increase, suggesting that the formation is saturable in these cells.
Ultimo aggiornamento 2012-04-10
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metabolisms šūnā un darbības mehānisms: nukleozīdu kināze intracelulāri metabolizē pirimidīna antimetabolītu gemcitabīnu (dfdc) par aktīviem difosfāta (dfdcdf) un trifosfāta (dfdctf) nukleozīdiem.
gemcitabine (dfdc), which is a pyrimidine antimetabolite, is metabolised intracellularly by nucleoside kinase to the active diphosphate (dfdcdp) and triphosphate (dfdctp) nucleosides.
Ultimo aggiornamento 2012-04-10
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