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diphenhydramin er rapporteret som værende en svag hæmmer af aldehyd oxidase i rotte lever, men det vides ikke, om det har en hæmmende virkning i leveren hos mennesker.
diphenhydramine is reported to be a weak inhibitor of aldehyde oxidase in rat liver, but its inhibitory effects in human liver are not known.
cimetidin, en ikke-specifik moderat inhibitor af flere leverenzymer, incl. både aldehyd oxidase og cyp3a4, bevirkede en 85% stigning i plasmakoncentrationen af zaleplon, fordi det hæmmede både de primære (aldehyd oxidase) og de sekundære (cyp3a4) enzymer, som er ansvarlige for metaboliseringen af zaleplon.
cimetidine, a non-specific moderate inhibitor of several hepatic enzymes including both aldehyde oxidase and cyp3a4, produced an 85% increase in plasma concentrations of zaleplon because it inhibited both the primary (aldehyde oxidase) and secondary (cyp3a4) enzymes responsible for zaleplon’s metabolism.