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the active substance in apoquel, oclacitinib, is an immunomodulator (a medicine that changes the activity of the immune system) that works by blocking the action of enzymes known as janus kinases.
apoqueli toimeaine oklatsitiniib on immunomodulaator (ravim, mis muudab immuunsüsteemi toimimist), mis blokeerib janus kinaasidena tuntud ensüümide toime.
by blocking the action of certain enzymes (called janus associated kinases), jakavi can reduce the size of the spleen in patients with myelofibrosis and relieve symptoms such as fever, night sweats, bone pain and weight loss in patients with myelofibrosis.
teatud ensüümide (neid nimetatakse janus kinaasideks) toime blokeerimise teel vähendab jakavi müelofibroosiga patsientidel põrna mõõtmeid ning leevendab müelofibroosiga patsientidel haiguse sümptomeid, nagu palavikku, öist higistamist, luuvalu ja kehakaalu langust.