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genotypically resistant

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arfgerðarónæmi

Laatste Update: 2017-04-26
Gebruiksfrequentie: 1
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Engels

treatment response is presented for the overall population (displayed by enfuvirtide use), and detailed by pi strata for the subgroup of patients with genotypically resistant strains in the table below.

IJslands

svörun við meðferð er sýnd fyrir allann hópinn (sýnt með notkun enfuvirtíð) og lýst með próteasahemli (pi strata) fyrir undirhóp sjúklinga með arfgerðarónæma stofna í töflunni hér að neðan.

Laatste Update: 2017-04-26
Gebruiksfrequentie: 1
Kwaliteit:

Engels

in healthy subjects who are genotypically poor metabolisers of cyp2d6 substrates (used as a surrogate for cyp2d6 inhibition), mean cmax and aucinf of a single 160 mg dose of a mirabegron ir formulation were 14% and 19% higher than in extensive metabolisers, indicating that cyp2d6 genetic polymorphism has minimal impact on the mean plasma exposure to mirabegron.

IJslands

hjá heilbrigðum einstaklingum sem vegna arfgerðar hafa lítil umbrot cyp2d6 hvarfefna (sem notuð eru sem staðgenglar fyrir cyp2d6 hömlun), voru meðalgildi cmax og aucinf eftir stakan 160 mg skammt af mirabegroni með tafarlausa losun 14% og 19% hærri en hjá þeim sem hafa mikil umbrot, sem sýnir að áhrif erfðafræðilegrar cyp2d6 fjölbreytni á meðalútsetningu fyrir mirabegroni í plasma eru í lágmarki.

Laatste Update: 2017-04-26
Gebruiksfrequentie: 1
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