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1'-hydroxymidazolam is metabolised predominantly by uridine diphosphate-glucuronosyltransferases (ugt) 2b4 and 2b7.
o 1 '- hidroximidazolam é metabolizado predominantemente pelas uridina difosfato glucuronosiltransferases (ugt) 2b4 e 2b7.
Laatste Update: 2011-10-23
Gebruiksfrequentie: 1
Kwaliteit:
Gelieve het te verwijderen indien je dit meent.
because 1'-hydroxymidazolam is an active metabolite, the sedative effect of midazolam may be increased and caution should be used when laropiprant is co-administered with midazolam.
como o 1 '- hidroximidazolam é um metabolito activo, pode ocorrer um aumento do efeito sedativo do midazolam pelo que se recomenda precaução quando o laropiprant é co- administrado com midazolam.
Laatste Update: 2011-10-23
Gebruiksfrequentie: 1
Kwaliteit:
Gelieve het te verwijderen indien je dit meent.
because 1'-hydroxymidazolam is an active metabolite, the sedative effect of midazolam may be increased and caution should be used when laropiprant is co-administered with midazolam.
como o 1 '- hidroximidazolam é um metabolito activo, pode ocorrer um aumento do efeito sedativo do midazolam pelo que se recomenda precaução quando o laropiprant é co- administrado com midazolam.
Laatste Update: 2012-04-12
Gebruiksfrequentie: 1
Kwaliteit:
co-administration of laropiprant 40 mg with midazolam increased the auc0-∞ and cmax of 1'-hydroxymidazolam, a midazolam metabolite, by 98% and 59%, respectively.
a co- administração de 40 mg de laropiprant com midazolam aumentou a auc0- ∞ e a cmáx do 1 '- hidroximidazolam, um metabolito do midazolam, em cerca de 98% e 59%, respectivamente.
Laatste Update: 2011-10-23
Gebruiksfrequentie: 1
Kwaliteit:
Gelieve het te verwijderen indien je dit meent.