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in base ai dati in vitro, il metabolismo dell’ azacitidina non appare mediato dagli isoenzimi del citocromo p450 (cyp), dalle udp-glucoronosiltransferasi (ugt), sulfotransferasi (sult) e glutatione transferasi (gst); le interazioni in vivo correlate a questi enzimi metabolizzanti sono pertanto considerate improbabili.
based on in vitro data, azacitidine metabolism does not appear to be mediated by cytochrome p450 isoenzymes (cyps), udp-glucuronosyltransferases (ugts), sulfotransferases (sults), and glutathione transferases (gsts); interactions related to these metabolizing enzymes in vivo are therefore considered unlikely.
最后更新: 2012-04-12
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