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[udp-glukuronyltransferas- substrat]
[udp-glucuronyl transferase substrate]
最后更新: 2017-04-26
使用频率: 1
质量:
mpa metaboliseras huvudsakligen av glukuronyltransferas till fenolglukuronid av mpa (mpag) som är farmakologiskt inaktiv.
mpa is metabolised principally by glucuronyl transferase to form the phenolic glucuronide of mpa (mpag), which is not pharmacologically active.
最后更新: 2012-04-11
使用频率: 2
质量:
1 '- hydroximidazolam metaboliseras huvudsakligen genom uridindifosfat- glukuronyltransferas (ugt) 2b4 och 2b7.
1'-hydroxymidazolam is metabolised predominantly by uridine diphosphate-glucuronosyltransferases (ugt) 2b4 and 2b7.
最后更新: 2011-10-23
使用频率: 1
质量:
potenta enzyminducerare som rifampicin, fenobarbital och fenytoin kan via effekt på udp - glukuronyltransferas minska plasmakoncentrationerna av abakavir något.
potent enzymatic inducers such as rifampicin, phenobarbital and phenytoin may via their action on udp-glucuronyltransferases slightly decrease the plasma concentrations of abacavir.
最后更新: 2012-04-11
使用频率: 2
质量:
abakavir metaboliseras via udp-glukuronyltransferas (ugt)-enzymer och alkoholdehydrogenas; samtidig administrering med inducerare eller hämmare av ugt-enzymer eller med substanser som elimineras via alkoholdehydrogenas kan påverka exponeringen av abakavir.
abacavir is metabolised by udp-glucuronyltransferase (ugt) enzymes and alcohol dehydrogenase; co-administration of inducers or inhibitors of ugt enzymes or with compounds eliminated through alcohol dehydrogenase could alter abacavir exposure.
最后更新: 2017-04-26
使用频率: 1
质量: