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in vitro, topotecano não inibiu as enzimas p450 humanas cyp1a2, cyp2a6, cyp2c8/ 9, cyp2c19, cyp2d6, cyp2e, cyp3a ou cyp4a, nem inibiu as enzimas citosólicas humanas di- hidropirimidina ou xantina- oxidase.
in vitro, topotécan n'a inhibé chez l'homme ni les enzymes p450 cyp1a2, cyp2a6, cyp2c8/ 9, cyp2c19, cyp2d6, cyp2e, cyp3a, ou cyp4a, ni les enzymes cytosoliques (la dihydropyrimidine ou la xanthine oxydase).