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tasimelteon 20 mg
tazimelteon 20 mg
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
tasimelteon is extensively metabolised.
tazimelteon se ekstenzivno metabolizira.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
the active substance is tasimelteon.
djelatna tvar je tazimelteon.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
hetlioz 20 mg hard capsules tasimelteon
hetlioz 20 mg tvrde kapsule tazimelteon
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
potential effect of alcohol on tasimelteon
mogući utjecaj alkohola na tazimelteon
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
each hard capsule contains 20 mg tasimelteon.
svaka tvrda kapsula sadrži 20 mg tazimelteona.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
each hard capsule contains 20 mg of tasimelteon.
svaka tvrda kapsula sadrži 20 mg tazimelteona.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
race does not affect apparent clearance of tasimelteon.
rasa ne utječe na prividni klirens tazimelteona.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
cyp2c19) in the metabolism of tasimelteon is unknown.
cyp2c19) u metabolizmu tazimelteona nije poznata.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
potential for other medicinal products to affect tasimelteon
mogućnost utjecaja drugih lijekova na tazimelteon
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
tasimelteon functions as a dmra at the mt1 and mt2 receptors.
tazimelteon djeluje kao dmra na receptorima mt1 i mt2.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
there are no data on the effects of tasimelteon on human fertility.
ne postoje podaci o učincima tazimelteona na plodnost u ljudi.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
it is unknown whether tasimelteon/metabolites are excreted in human milk.
nije poznato izlučuje li se tazimelteon/metaboliti u majčino mlijeko u ljudi.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
tasimelteon exhibits a greater affinity for the mt2 as compared to the mt1 receptor.
tazimelteon pokazuje veći afinitet za receptore mt2 u odnosu na receptore mt1.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
cyp1a2 and cyp3a4 are enzymes identified to play a role in the metabolism of tasimelteon.
cyp1a2 i cyp3a4 su enzimi za koje je utvrđeno da imaju ulogu u metabolizmu tazimelteona.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
as a precautionary measure, it is preferable to avoid the use of tasimelteon during pregnancy.
kao mjera opreza, preporučuje se izbjegavanje uporabe tazimelteona tijekom trudnoće.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
major metabolites had 13-fold or less activity at melatonin receptors compared to tasimelteon.
glavni metaboliti imali su najmanje 13 puta manju aktivnost na receptorima melatonina u usporedbi s tazimelteonom.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
medicinal products that inhibit cyp1a2 and cyp3a4 have been shown to alter the metabolism of tasimelteon in vivo.
pokazalo se da lijekovi koji inhibiraju cyp1a2 i cyp3a4 mijenjaju metabolizam tazimelteona in vivo.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
in pregnant rats administered tasimelteon during the period of organogenesis, there were no effects on embryofoetal development.
u gravidnih štakora koji su tijekom organogeneze primali tazimelteon nije bilo utjecaja na embriofetalni razvoj.
Last Update: 2017-04-26
Usage Frequency: 1
Quality:
adverse reactions leading to discontinuation occurred in 2.3% of tasimelteon-treated patients.
nuspojave koje su rezultirale prekidom uporabe lijeka zabilježene su kod 2,3 % bolesnika liječenih tazimelteonom.
Last Update: 2017-04-26
Usage Frequency: 1
Quality: