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cl channels
canais de cloreto
Last Update: 2014-12-09
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moxidectin interacts with gaba and glutamate- gated chloride channels.
a moxidectina interage com os canais de cloro controlados pelo gaba e pelo glutamato.
Last Update: 2017-04-26
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sarolaner blocks gaba- and glutamate-gated chloride channels in the central nervous system of insects and acarines.
sarolaner bloqueia os canais de cloro-ligantes recetores gaba e glutamato no sistema nervoso central dos insetos e acarídeos.
Last Update: 2017-04-26
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compounds of the class bind selectively and with high affinity to glutamate-gated chloride ion channels which occur in invertebrate nerve or muscle cells.
os compostos da classe ligam-se selectivamente e com uma afinidade muito elevada aos canais de iões de cloro com terminais glutamato, que se encontram nas células nervosas e musculares dos invertebrados.
Last Update: 2017-04-26
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disruption of these receptors by sarolaner prevents the uptake of chloride ions by gaba and glutamate gated ion channels, thus resulting in increased nerve stimulation and death of the target parasite.
a rutura destes recetores pelo sarolaner impede a transferência dos iões cloro pelos canais de cloro-ligantes recetores gaba e glutamato, resultando num aumento da estimulação nervosa e morte dos parasitas alvo.
Last Update: 2017-04-26
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moxidectin interferes with different receptors (gaba and glutamate-gated chloride channels) in the other parasites, leading to their paralysis, death and expulsion.
a moxidectina interfere com diferentes receptores (canais de cloro controlados pelo gaba e pelo glutamato) nos outros parasitas, o que leva à sua paralisia, morte e expulsão.
Last Update: 2012-04-12
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milbemycin oxime, like avermectins and other milbemycins, increases nematode and insect membrane permeability to chloride ions via glutamate-gated chloride ion channels (related to vertebrate gaba and glycine receptors).
a milbemicina oxima, como avermectinas e outras milbemicinas, aumenta a permeabilidade do nemátodo e da membrana do insecto a iões de cloro através de canais de iões de glutamato (relacionados com receptores gaba vertebrados e de glicina).
Last Update: 2017-04-26
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