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poliglutamāta formas paliek šūnā un ir pat vēl spēcīgāki ts un garft inhibitori.
polyglutamatformerne forbliver i cellerne og fungerer som endnu mere potente hæmmere af ts og garft.
Last Update: 2011-10-23
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Šūnā enzīma folipoliglutamāta sintetāzes ietekmē pemetrekseds tiek ātri un efektīvi pārvērsts par poliglutamāta formām.
når pemetrexed er trængt ind i cellen, omdannes det hurtigt til polyglutamatformer via enzymfolylpolyglutamatsyntetase.
Last Update: 2012-04-11
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