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interaktioner som medieras av effekter på transportörer
interactions mediated by effects on transporters
Last Update: 2017-04-26
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leverupptaget av simeprevir medieras av oatp1b1/3.
hepatic uptake of simeprevir is mediated by oatp1b1/3.
Last Update: 2017-04-26
Usage Frequency: 1
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aktiv renal sekretion medieras av oct2-transportör.
active renal secretion is mediated via oct2 transporter.
Last Update: 2017-04-26
Usage Frequency: 1
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metabolismen av celecoxib medieras primärt via cytokrom p450cyp2c9.
celecoxib metabolism is primarily mediated via cytochrome p450 cyp2c9.
Last Update: 2017-04-26
Usage Frequency: 3
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metabolismen av melatonin medieras företrädesvis av cyp1a-enzymer.
melatonin’s metabolism is mainly mediated by cyp1a enzymes.
Last Update: 2017-04-26
Usage Frequency: 2
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metabolismen av den här aktiva metaboliten medieras också av cyp3a4.
the metabolism of this active metabolite also involves cyp3a4.
Last Update: 2017-04-26
Usage Frequency: 3
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man antar att dessa effekter medieras av mtp-hämning på enterocytnivå.
it is assumed that these effects are mediated by mtp inhibition at the level of the enterocyte.
Last Update: 2017-04-26
Usage Frequency: 3
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darifenacins metabolism hos långsamma cyp2d6-metaboliserare medieras huvudsakligen av cyp3a4.
the metabolism of darifenacin in cyp2d6 poor metabolisers is principally mediated by cyp3a4.
Last Update: 2017-04-26
Usage Frequency: 1
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in vitro medieras den här vägen av cyp3a4, cyp2c19, cyp1a2 och cyp2b6.
in vitro, this metabolic pathway is mediated by cyp3a4, cyp2c19, cyp1a2 and cyp2b6.
Last Update: 2017-04-26
Usage Frequency: 1
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det är därför möjligt att läkemedelsinteraktioner kan uppträda, vilka medieras genom hämning av transportproteiner.
there is thus the potential of drug interactions mediated by inhibition of transporters.
Last Update: 2012-04-11
Usage Frequency: 2
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nikotinsyrainducerad flush medieras huvudsakligen genom frisättning av prostaglandin d2 (pgd2) i huden.
nicotinic acid-induced flushing is mediated primarily by release of prostaglandin d2 (pgd2) in the skin.
Last Update: 2017-04-26
Usage Frequency: 1
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bildningen av treohydrobupropion har däremot rapporterats i litteraturen att medieras med 11-beta-hydroxisteroiddehydrogenas 1.
in contrast, formation of threohydrobupropion has been reported in the literature to be mediated by 11-beta-hydroxysteroid dehydrogenase 1.
Last Update: 2017-04-26
Usage Frequency: 1
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lasofoxifen är ett serm-medel, vars biologiska effekt i stor utsträckning medieras genom bindning till östrogenreceptorer.
lasofoxifene is a serm whose biological actions are largely mediated through binding to estrogen receptors.
Last Update: 2017-04-26
Usage Frequency: 3
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9 laropiprant verkningsmekanism nikotinsyrainducerad flush medieras huvudsakligen genom frisättning av prostaglandin d2 (pgd2) i huden.
10 laropiprant mechanism of action nicotinic acid-induced flushing is mediated primarily by release of prostaglandin d2 (pgd2) in the skin.
Last Update: 2012-04-11
Usage Frequency: 4
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den antikoagulerande aktiviteten medieras via antitrombin iii (atiii), vilket resulterar i antitrombotisk effekt hos människa.
the antithrombotic activity is mediated by antithrombin iii (atiii), resulting in human antithrombotic effect.
Last Update: 2017-04-26
Usage Frequency: 1
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saxagliptin: metabolismen av saxagliptin medieras primärt av cytokrom p450 3a4/5 (cyp3a4/5).
saxagliptin: the biotransformation of saxagliptin is primarily mediated by cytochrome p450 3a4/5 (cyp3a4/5).
Last Update: 2017-04-26
Usage Frequency: 1
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cytokrom (cyp) 450-medierade metaboliska läkemedelsinteraktioner förväntas inte eftersom decitabins metabolism inte medieras via detta system utan genom oxidativ deaminering.
cytochrome (cyp) 450-mediated metabolic interactions are not anticipated as decitabine metabolism is not mediated by this system but by oxidative deamination.
Last Update: 2017-04-26
Usage Frequency: 1
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tnfα (tumörnekrosfaktor alfa) medierar inflammation och modulerar det cellulära immunsvaret.
tumour necrosis factor alpha (tnfα) mediates inflammation and modulates cellular immune responses.
Last Update: 2017-04-26
Usage Frequency: 3
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