Results for plasmamelatoninhalter translation from Swedish to English

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Swedish

försiktighet måste iakttas för patienter som behandlas med cimetidin, en cyp2d-hämmare, som ger höjda plasmamelatoninhalter genom att hämma metabolismen av melatonin.

English

caution should be exercised in patients on cimetidine a cyp2d inhibitor, which increases plasma melatonin levels, by inhibiting its metabolism.

Last Update: 2017-04-26
Usage Frequency: 2
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Swedish

kombinationen bör undvikas. • försiktighet måste iakttas för patienter som behandlas med 5 - eller 8- metoxipsoralen (5 - och 8- mop), vilket ökar melatoninhalterna genom att hämma metabolismen av melatonin. • försiktighet måste iakttas för patienter som behandlas med cimetidin, en cyp2d - hämmare, som ger höjda plasmamelatoninhalter genom att hämma metabolismen av melatonin. • cigarettrökning kan sänka melatoninhalterna genom en induktion av cyp1a2. • försiktighet måste iakttas för patienter som behandlas med östrogener (t. ex. hormonella preventivmedel eller hormonell substitutionsbehandling), vilka ökar melatoninhalterna genom att hämma metabolismen av melatonin med cyp1a1 och cyp1a2. • cyp1a2- hämmare, som kinoloner, kan orsaka en ökad melatoninexponering. • cyp1a2- inducerare, såsom karbamazepin och rifampicin, kan ge upphov till reducerade plasmakoncentrationer av melatonin. • det finns även omfattande data i litteraturen avseende effekten på den endogena melatonininsöndringen från adrenerga agonister/ antagonister, opiatagonister/ antagonister, antidepressiva läkemedel, prostaglandinhämmare, bensodiazepiner, tryptofan och alkohol.

English

the combination should be avoided. • caution should be exercised in patients on 5- or 8-methoxypsoralen (5 and 8-mop), which increases melatonin levels by inhibiting its metabolism. • caution should be exercised in patients on cimetidine a cyp2d inhibitor, which increases plasma melatonin levels, by inhibiting its metabolism. • cigarette smoking may decrease melantonin levels due to induction of cyp1a2. • caution should be exercised in patients on oestrogens (e. g. contraceptive or hormone replacement therapy), which increase melatonin levels by inhibiting its metabolism by cyp1a1 and cyp1a2. • cyp1a2 inhibitors such as quinolones may give rise to increased melatonin exposure. • cyp1a2 inducers such as carbamazepine and rifampicin may give rise to reduced plasma concentrations of melatonin. • there is a large amount of data in the literature regarding the effect of adrenergic agonists/ antagonists, opiate agonists/ antagonists, antidepressant medicinal products, prostaglandin inhibitors, benzodiazepines, tryptophan and alcohol, on endogenous melatonin secretion.

Last Update: 2011-10-23
Usage Frequency: 1
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